SCHEMBL14969291

SCHEMBL14969291

O=Cc1ccc(-c2ccc(F)nc2)cc1F

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 5/20 0.46
CYP11B2 P19099 2/20 0.43
CYP2E1 P05181 1/20 0.42
CYP2A6 P11509 1/20 0.42
CYP2B6 P20813 1/20 0.42
GRIN1 Q05586 1/20 0.39
GRIN2B Q13224 1/20 0.39
PIK3CD O00329 1/20 0.39
ABL1 P00519 1/20 0.39
EGFR P00533 1/20 0.39
HCK P08631 1/20 0.39
SRC P12931 1/20 0.39
KDR P35968 1/20 0.39
PIK3CA P42336 1/20 0.39
PIK3CB P42338 1/20 0.39
MTOR P42345 1/20 0.39
PIK3CG P48736 1/20 0.39
EPHB4 P54760 1/20 0.39
PRKDC P78527 1/20 0.39
DHODH Q02127 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18003520 0.81 PIK3CA (0.50) ERN1PIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL14968263 0.81 ERN1 (0.43) ERN1CYP11B2CYP2E1CYP2A6CYP2B6
SCHEMBL29828302 0.79 ERN1 (0.46) ERN1ESR1ESR2
SCHEMBL21199864 0.77 ERN1 (0.45) ERN1CYP11B2CYP11B1ESR1ESR2
SCHEMBL4735387 0.76 ERN1 (0.51) ERN1MAPT
SCHEMBL17832843 0.76 ERN1 (0.40) ERN1PIK3CDABL1EGFRHCK
SCHEMBL2774294 0.76 KIF11 (0.44) ERN1ESR1ESR2MAPT
SCHEMBL15903722 0.76 ALDH1A1 (0.35)
SCHEMBL23905206 0.75 ERN1 (0.52) ERN1EGFRPIK3CAPIK3CG
SCHEMBL15645548 0.75 ERN1 (0.46) ERN1CYP11B2CYP2E1CYP2A6CYP2B6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013074387-A1 IMIDAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2013-05-23 WO disclosed
WO-2013074387-A1 IMIDAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2013-05-23 WO disclosed