SCHEMBL14968263

SCHEMBL14968263

O=Cc1c(F)cc(-c2ccc(F)nc2)cc1F

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 5/20 0.43
CYP2A6 P11509 3/20 0.43
CYP2B6 P20813 3/20 0.43
CYP2E1 P05181 1/20 0.43
CYP11B2 P19099 2/20 0.41
PDE3B Q13370 1/20 0.38
PDE3A Q14432 1/20 0.38
MAPT P10636 2/20 0.38
GRIA2 P42262 2/20 0.37
GRIN1 Q05586 1/20 0.37
GRIN2B Q13224 1/20 0.37
DHODH Q02127 1/20 0.37
CYP3A4 P08684 2/20 0.37
CYP2C19 P33261 2/20 0.37
JAK2 O60674 1/20 0.36
RET P07949 1/20 0.36
KDR P35968 1/20 0.36
GSK3A P49840 1/20 0.36
RPS6KA3 P51812 1/20 0.36
LIMK1 P53667 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20456821 0.81 ERN1 (0.41) ERN1KDR
SCHEMBL14969291 0.81 ERN1 (0.46) ERN1CYP2A6CYP2B6CYP2E1CYP11B2
SCHEMBL20456786 0.76 ERN1 (0.39) ERN1PDE3BPDE3AKDR
SCHEMBL26104326 0.76 CYP2A6 (0.64) CYP2A6CYP2B6CYP2E1CYP11B2MAPT
SCHEMBL14879555 0.72 AHR (0.43) ERN1
SCHEMBL13083660 0.72 PTGS2 (0.43) ERN1CYP2A6MAPTCYP2C19RPS6KA3
SCHEMBL27422573 0.71 CYP2A6 (0.40) CYP2A6CYP2B6CYP2E1CYP11B2PDE3B
SCHEMBL22657759 0.71 AKR1C2 (0.47) ERN1CYP2A6
SCHEMBL31207438 0.70 ALDH1A1 (0.48) CYP2A6CYP2B6CYP2E1CYP11B2PDE3B
SCHEMBL20456721 0.70 TGFBR1 (0.36) ERN1KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013074387-A1 IMIDAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2013-05-23 WO disclosed