SCHEMBL14972766

SCHEMBL14972766

O=C1OC=CC1=CNCc1cccnc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.46
CYP2D6 P10635 1/20 0.46
LMNA P02545 1/20 0.42
RECQL P46063 1/20 0.42
CTSL P07711 1/20 0.41
ALDH1A1 P00352 3/20 0.41
LTA4H P09960 1/20 0.41
USP2 O75604 1/20 0.41
POLB P06746 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
KDM4E B2RXH2 1/20 0.40
PKM P14618 1/20 0.40
CHRM2 P08172 1/20 0.40
MAPT P10636 1/20 0.40
NPSR1 Q6W5P4 1/20 0.39
FES P07332 1/20 0.39
RET P07949 1/20 0.39
MARK3 P27448 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7547160 0.77 CYP1A2 (0.45) CYP1A2CYP2D6LMNARECQLALDH1A1
SCHEMBL7547164 0.77 CYP1A2 (0.45) CYP1A2CYP2D6LMNARECQLALDH1A1
SCHEMBL1310957 0.75 KMT2A (0.38) LMNAALDH1A1POLBL3MBTL1CHRM2
SCHEMBL1310330 0.75 SMN1; SMN2 (0.39) LMNAALDH1A1USP2POLBL3MBTL1
SCHEMBL1310266 0.72 ALDH1A1 (0.52) ALDH1A1USP2POLBNPC1RAB9A
SCHEMBL348709 0.72 CYP1A2 (0.68) CYP1A2CYP2D6LMNARECQLALDH1A1
SCHEMBL14972765 0.71 CYP1A2 (0.45) CYP1A2CYP2D6LMNARECQLALDH1A1
SCHEMBL3160679 0.69 CYP1A2 (0.62) CYP1A2CYP2D6LMNARECQLCTSL
SCHEMBL26780009 0.69 CYP1A2 (0.62) CYP1A2CYP2D6LMNARECQLCTSL
SCHEMBL15065573 0.66 CYP1A2 (0.58) CYP1A2CYP2D6LMNARECQLCTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8846125-B2 Enaminocarbonyl compounds and their use INSTYTUT CHEMII ORGANICZNEJ, POLSKA AKADEMIA NAUK (PL) 2014-09-30 US claimed
EP-2391614-B1 ENAMINOCARBONYL COMPOUNDS AND THEIR USE INST CHEMII ORGANICZNEJ POLSKA AKADEMIA NAUK (PL) 2013-05-29 EP claimed
EP-2391614-B1 ENAMINOCARBONYL COMPOUNDS AND THEIR USE INST CHEMII ORGANICZNEJ POLSKA AKADEMIA NAUK (PL) 2013-05-29 EP disclosed