SCHEMBL14972765

SCHEMBL14972765

O=C1OCCC1=CNCc1cccnc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.45
CYP2D6 P10635 1/20 0.45
HSP90AA1 P07900 1/20 0.44
HSP90AB1 P08238 1/20 0.44
ALDH1A1 P00352 3/20 0.43
KDM4E B2RXH2 2/20 0.43
PKM P14618 1/20 0.43
KMT2A Q03164 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.42
LMNA P02545 1/20 0.41
RECQL P46063 1/20 0.41
HSD17B10 Q99714 1/20 0.41
GAA P10253 1/20 0.40
MAPT P10636 1/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
USP2 O75604 1/20 0.40
POLB P06746 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
LTA4H P09960 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1310500 0.83 KMT2A (0.60) HSP90AA1HSP90AB1ALDH1A1KMT2ASMN1; SMN2
SCHEMBL1310955 0.76 KMT2A (0.49) HSP90AA1HSP90AB1ALDH1A1KMT2ASMN1; SMN2
SCHEMBL1310328 0.76 KMT2A (0.55) HSP90AA1HSP90AB1ALDH1A1KDM4EKMT2A
SCHEMBL14972763 0.74 KMT2A (0.66) HSP90AA1HSP90AB1ALDH1A1KMT2ASMN1; SMN2
SCHEMBL14972752 0.74 HSP90AA1 (0.49) HSP90AA1HSP90AB1ALDH1A1KDM4EKMT2A
SCHEMBL1310264 0.73 ALDH1A1 (0.65) HSP90AA1HSP90AB1ALDH1A1KDM4EKMT2A
SCHEMBL1325020 0.71 HSP90AA1 (0.49) HSP90AA1HSP90AB1ALDH1A1KMT2ARECQL
SCHEMBL1311593 0.71 HSP90AA1 (0.56) HSP90AA1HSP90AB1ALDH1A1PKMKMT2A
SCHEMBL14972766 0.71 CYP1A2 (0.46) CYP1A2CYP2D6ALDH1A1KDM4EPKM
SCHEMBL348709 0.71 CYP1A2 (0.68) CYP1A2CYP2D6ALDH1A1KDM4EPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8846125-B2 Enaminocarbonyl compounds and their use INSTYTUT CHEMII ORGANICZNEJ, POLSKA AKADEMIA NAUK (PL) 2014-09-30 US claimed
EP-2391614-B1 ENAMINOCARBONYL COMPOUNDS AND THEIR USE INST CHEMII ORGANICZNEJ POLSKA AKADEMIA NAUK (PL) 2013-05-29 EP claimed
EP-2391614-B1 ENAMINOCARBONYL COMPOUNDS AND THEIR USE INST CHEMII ORGANICZNEJ POLSKA AKADEMIA NAUK (PL) 2013-05-29 EP disclosed