SCHEMBL14977339

SCHEMBL14977339

CNC(=O)c1c(-c2ccc(F)cc2)nc2sc(-c3cc(C(=O)NC(C)(C)c4ccccc4)ccc3OC)cn12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 1/20 0.43
ROCK1 Q13464 1/20 0.43
HDAC6 Q9UBN7 1/20 0.38
PPARG P37231 1/20 0.37
PTGDR2 Q9Y5Y4 3/20 0.36
TP53 P04637 3/20 0.36
MAPT P10636 1/20 0.36
LMNA P02545 2/20 0.35
KIT P10721 1/20 0.35
MEN1 O00255 1/20 0.34
NPC1 O15118 1/20 0.34
KMT2A Q03164 1/20 0.34
POLB P06746 1/20 0.34
DGAT2 Q96PD7 1/20 0.34
HSP90AA1 P07900 1/20 0.34
TUBB4A P04350 1/20 0.34
TUBB P07437 1/20 0.34
TUBA3C P0DPH7 1/20 0.34
TUBA1B P68363 1/20 0.34
TUBA4A P68366 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14977379 0.90 DGAT2 (0.42) ROCK2ROCK1PPARGPTGDR2TP53
SCHEMBL14977707 0.90 PPARG (0.39) ROCK2ROCK1PPARGPTGDR2MAPT
SCHEMBL14977623 0.88 PPARG (0.39) ROCK2ROCK1PPARGPTGDR2TP53
SCHEMBL14977301 0.87 CSNK1D (0.36) ROCK2ROCK1PTGDR2TP53MAPT
SCHEMBL14977718 0.87 ROCK2 (0.35) ROCK2ROCK1PTGDR2TP53MAPT
SCHEMBL14977224 0.86 KIT (0.39) PPARGPTGDR2MAPTLMNAKIT
SCHEMBL2466314 0.86 ROCK2 (0.44) ROCK2ROCK1PPARGNPC1DGAT2
SCHEMBL14977778 0.86 ROCK2 (0.39) ROCK2PTGDR2MAPTMEN1NPC1
SCHEMBL14977569 0.86 MAPK14 (0.37) PPARGMAPTDGAT2
SCHEMBL14986300 0.85 HDAC6 (0.41) HDAC6PTGDR2TP53MAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013075173-A1 COMPOUNDS FOR THE TREATMENT OF HCV BIOTA SCIENTIFIC MANAGEMENT PTY LTD (AU) 2013-05-30 WO disclosed
WO-2013075173-A1 COMPOUNDS FOR THE TREATMENT OF HCV BIOTA SCIENTIFIC MANAGEMENT PTY LTD (AU) 2013-05-30 WO disclosed