SCHEMBL1497962

SCHEMBL1497962

COC(C)n1ncc(N)c1N

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5425218 0.81
SCHEMBL144678 0.79 PIK3CD (0.30)
SCHEMBL4730392 0.77
SCHEMBL5424987 0.76 HCAR3 (0.34)
SCHEMBL94060 0.75
SCHEMBL14321038 0.75
SCHEMBL5160602 0.73
SCHEMBL5429996 0.73
SCHEMBL5393771 0.72 L3MBTL1 (0.34)
SCHEMBL5423902 0.71 TLR7 (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 100 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025129303-A1 METHODS FOR TREATING KERATIN FIBERS WITH OSMOLYTES, CARBOXYLIC ACIDS AND AMINO ACIDS L'OREAL (FR) 2025-06-26 WO disclosed
EP-4362902-A1 COMPOSITIONS CONTAINING DIRECT DYES FOR IMPARTING COLOR AND TONE TO THE HAIR L'OREAL (FR) 2024-05-08 EP disclosed
EP-4362891-A1 COMPOSITION COMPRISING AT LEAST ONE PARTICULAR COUPLER, AT LEAST ONE PARTICULAR OXIDATION BASE, AT LEAST ONE FATTY SUBSTANCE AND AT LEAST ONE ANIONIC POLYSACCHARIDE L'OREAL (FR) 2024-05-08 EP disclosed
EP-4362889-A1 COMPOSITION COMPRISING AT LEAST ONE OXIDATION DYE, 1,3-PROPANEDIOL, AT LEAST ONE ALKALINE AGENT AND AT LEAST ONE FATTY SUBSTANCE L'OREAL (FR) 2024-05-08 EP disclosed
EP-4362906-A1 COMPOSITION COMPRISING SHEA, AN ALKYL(POLY)GLYCOSIDE, A POLYSACCHARIDE AND A DYE L'OREAL (FR) 2024-05-08 EP disclosed
CN-113795435-B Soluble package of pre-measured powdered hair bleach 莱雅公司 2023-04-25 CN disclosed
WO-2023275168-A1 COMPOSITION COMPRISING AT LEAST ONE PARTICULAR COUPLER, AT LEAST ONE PARTICULAR OXIDATION BASE, AT LEAST ONE FATTY SUBSTANCE AND AT LEAST ONE ANIONIC POLYSACCHARIDE L'OREAL (FR) 2023-01-05 WO disclosed
WO-2023278726-A1 COMPOSITIONS CONTAINING DIRECT DYES FOR IMPARTING COLOR AND TONE TO THE HAIR L'OREAL (FR) 2023-01-05 WO disclosed
WO-2023275193-A1 COMPOSITION COMPRISING AT LEAST ONE OXIDATION DYE, 1,3-PROPANEDIOL, AT LEAST ONE ALKALINE AGENT AND AT LEAST ONE FATTY SUBSTANCE L'OREAL (FR) 2023-01-05 WO disclosed
WO-2023275187-A1 COMPOSITION COMPRISING SHEA, AN ALKYL(POLY)GLYCOSIDE, A POLYSACCHARIDE AND A DYE L'OREAL (FR) 2023-01-05 WO disclosed
WO-2012059407-A1 FOAM DYE COMPOSITION COMPRISING A MONOSACCHARIDE OR DISACCHARIDE L'OREAL (FR) 2012-05-10 WO disclosed
WO-2011157699-A2 METHOD FOR LIGHTENING OR DYEING IN THE PRESENCE OF AMMONIUM (BI)CARBONATE AND A BASE, AND DEVICE L'OREAL (FR) 2011-12-22 WO disclosed
WO-2011076647-A2 INVERSE EMULSION FOR TREATING THE HAIR COMPRISING A PARTICULAR FATTY SUBSTANCE AND AN ALKALINE AGENT L'OREAL (FR) 2011-06-30 WO disclosed
WO-2011076646-A2 AGENT FOR DYEING AND/OR BLEACHING KERATIN FIBRES, COMPRISING AN INVERSE EMULSION COMPRISING AN OXIDIZING AGENT L'OREAL (FR) 2011-06-30 WO disclosed
WO-2011076792-A1 AGENT FOR DYEING AND/OR BLEACHING KERATINOUS FIBRES IN TWO OR MORE PARTS IN THE FORM OF AN EMULSION AND OF A DISPERSION L'OREAL (FR) 2011-06-30 WO disclosed
WO-2011076672-A2 AGENT FOR DYEING AND/OR BLEACHING KERATINOUS FIBRES IN TWO OR MORE PARTS, COMPRISING AN ALKALINE COMPOSITION IN AN INVERSE EMULSION L'OREAL (FR) 2011-06-30 WO disclosed
WO-2011027077-A2 COMPOSITION COMPRISING A HYDROPHOBIC DYE, A SPECIFIC MINERAL AND/OR ORGANIC ALKALINE AGENT, A SPECIFIC COMPOUND (I) AND A SPECIFIC ORGANIC COMPOUND (II), AND USE THEREOF IN DYEING L'OREAL (FR) 2011-03-10 WO disclosed
WO-2011027076-A2 DYEING METHOD CONSISTING IN APPLYING A METALLIC SALT AND A COMPOSITION CONTAINING A HYDROPHOBIC DYE AND A SPECIFIC COMPOUND L'OREAL (FR) 2011-03-10 WO disclosed
EP-1586303-A1 Dye composition comprising at least one diaminopyrazole as oxidation base and at least one 6-alkoxy-2,3-diaminopyridine as coupler L'OREAL (FR) 2005-10-19 EP disclosed
EP-1457198-A1 Dyeing composition comprising at least one diaminopyrazole precursor and at least one 6-alcoxy 2,3-diaminopyridine coupler L'OREAL (FR) 2004-09-15 EP disclosed