SCHEMBL14980754

SCHEMBL14980754

CCCN1CCC=C(c2ccc(C)c(N)c2)C1

nearest known ligand 0.51

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 1/20 0.51
CHRM4 P08173 1/20 0.51
CHRM5 P08912 1/20 0.51
ADRA2A P08913 1/20 0.51
ADRA2B P18089 1/20 0.51
ADRA2C P18825 1/20 0.51
CHRM3 P20309 1/20 0.51
KCNH2 Q12809 1/20 0.51
TMEM97 Q5BJF2 1/20 0.51
SIGMAR1 Q99720 1/20 0.51
INSR P06213 1/20 0.41
IGF1R P08069 1/20 0.41
MAPK8 P45983 1/20 0.41
ALK Q9UM73 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2207458 0.89 CHRM2 (0.51) CHRM2CHRM4CHRM5ADRA2AADRA2B
SCHEMBL2205877 0.83 CHRM2 (0.46) CHRM2CHRM4CHRM5ADRA2AADRA2B
SCHEMBL2204492 0.81 ALDH1A1 (0.46) CHRM2CHRM4CHRM5ADRA2AADRA2B
Bromide SCHEMBL11203229 0.77 CHRM2 (0.49) CHRM2CHRM4CHRM5ADRA2AADRA2B
SCHEMBL2207405 0.76 CHRM2 (0.47) CHRM2CHRM4CHRM5ADRA2AADRA2B
SCHEMBL11196119 0.76 IGF1R (0.49) CHRM2CHRM4CHRM5ADRA2AADRA2B
SCHEMBL11198460 0.74 DRD2 (0.49) CHRM2CHRM4CHRM5ADRA2AADRA2B
Hydrochloric Acid SCHEMBL11199175 0.73 DRD2 (0.48) CHRM2CHRM4CHRM5ADRA2AADRA2B
SCHEMBL11198743 0.72 DRD2 (0.52) CHRM2CHRM4CHRM5ADRA2AADRA2B
SCHEMBL11260900 0.71 DRD2 (0.50) CHRM2CHRM4CHRM5ADRA2AADRA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2188292-B1 2- [ (2-{PHENYLAMINO}-1H-PYRROLO [2, 3-D]PYRIMIDIN-4-YL) AMINO]BENZAMIDE DERIVATIVES AS IGF-1R INHIBITORS FOR THE TREATMENT OF CANCER GLAXOSMITHKLINE IP DEV LTD (GB) 2013-05-29 EP disclosed