SCHEMBL15012018

SCHEMBL15012018

COCCCOc1cccc(COc2ccc(CNC3CC3)cc2)c1

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.50
MAOB P27338 3/20 0.46
HRH3 Q9Y5N1 2/20 0.45
BCHE P06276 3/20 0.44
CYP2C9 P11712 1/20 0.43
KMT2A Q03164 3/20 0.43
KDM4E B2RXH2 3/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
ENPP2 Q13822 1/20 0.43
MEN1 O00255 2/20 0.42
KDM1A O60341 2/20 0.42
FFAR1 O14842 1/20 0.42
FOXM1 Q08050 1/20 0.42
NPC1 O15118 1/20 0.41
LMNA P02545 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL695510 0.89 ALDH1A1 (0.62) ALDH1A1MAOBKDM4EKDM1A
SCHEMBL2807484 0.83 KMT2A (0.47) ALDH1A1MAOBHRH3BCHECYP2C9
SCHEMBL15012151 0.80 MEN1 (0.42) ALDH1A1MAOBBCHEKMT2AKDM4E
SCHEMBL5555860 0.77 BCHE (0.65) BCHEKMT2AKDM4ESMN1; SMN2MEN1
SCHEMBL15012179 0.76 KDM4E (0.48) ALDH1A1MAOBBCHEKMT2AKDM4E
SCHEMBL8265518 0.75 CNR1 (0.55) ALDH1A1KDM4E
SCHEMBL5555203 0.75 HRH3 (0.58) ALDH1A1HRH3CYP2C9KMT2AKDM4E
Ammonia Solution, Strong SCHEMBL9637696 0.75 ALDH1A1 (0.59) ALDH1A1CYP2C9KDM4EKDM1A
SCHEMBL9637698 0.75 ALDH1A1 (0.56) ALDH1A1HRH3CYP2C9KDM1A
SCHEMBL89233 0.75 ALDH1A1 (0.66) ALDH1A1HRH3KMT2AKDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013084241-A1 COMPOUNDS AS INHIBITORS OF RENIN CADILA HEALTHCARE LIMITED (IN) 2013-06-13 WO disclosed