Triamcinolone

Triamcinolone

SCHEMBL1502196

C[C@]12C=CC(=O)C=C1CC[C@H]1[C@@H]3C[C@@H](O)[C@](O)(C(=O)CO)[C@@]3(C)CC(O)C12F

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

NR3C1

The experimentally established mechanism targets of Triamcinolone. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR3C1 known ✓ P04150 9/20 1.00
HIF1A Q16665 8/20 1.00
CYP3A4 P08684 7/20 1.00
LMNA P02545 5/20 1.00
HSD17B10 Q99714 4/20 1.00
PGR P06401 4/20 1.00
NFKB1 P19838 3/20 1.00
CYP2C9 P11712 3/20 1.00
PMP22 Q01453 2/20 1.00
CYP2J2 P51589 1/20 1.00
BLM P54132 1/20 1.00
CYP2C19 P33261 1/20 1.00
TSHR P16473 2/20 0.86
AR P10275 2/20 0.86
MEN1 O00255 1/20 0.86
CYP2D6 P10635 1/20 0.86
KMT2A Q03164 1/20 0.86
APEX1 P27695 1/20 0.86
NPSR1 Q6W5P4 1/20 0.86
IKBKB O14920 1/20 0.86

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Triamcinolone SCHEMBL1884154 1.00 NR3C1 (1.00) NR3C1HIF1ACYP3A4LMNAHSD17B10
Triamcinolone SCHEMBL9863653 1.00 NR3C1 (1.00) NR3C1HIF1ACYP3A4LMNAHSD17B10
Triamcinolone SCHEMBL601461 1.00 NR3C1 (1.00) NR3C1HIF1ACYP3A4LMNAHSD17B10
Triamcinolone SCHEMBL14373318 1.00 NR3C1 (1.00) NR3C1HIF1ACYP3A4LMNAHSD17B10
Triamcinolone SCHEMBL8813577 1.00 NR3C1 (1.00) NR3C1HIF1ACYP3A4LMNAHSD17B10
Triamcinolone SCHEMBL24622562 1.00 NR3C1 (1.00) NR3C1HIF1ACYP3A4LMNAHSD17B10
Triamcinolone SCHEMBL601462 1.00 NR3C1 (1.00) NR3C1HIF1ACYP3A4LMNAHSD17B10
Triamcinolone SCHEMBL570639 1.00 NR3C1 (1.00) NR3C1HIF1ACYP3A4LMNAHSD17B10
Triamcinolone SCHEMBL22962813 1.00 NR3C1 (1.00) NR3C1HIF1ACYP3A4LMNAHSD17B10
Triamcinolone SCHEMBL4447 1.00 NR3C1 (1.00) NR3C1HIF1ACYP3A4LMNAHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 20 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1143950-B1 TOPICAL APPLICATION PRODUCTS AGAINST ONYCHOMYCOSES BIOEQUAL AG (CH) 2005-03-09 EP claimed
EP-1143950-A3 TOPICAL APPLICATION PRODUCTS IPR-Institute for Pharmaceutical Research AG (CH) 2002-05-15 EP claimed
EP-1143950-A2 TOPICAL APPLICATION PRODUCTS IPR-Institute for Pharmaceutical Research AG (CH) 2001-10-17 EP claimed
WO-2000015202-A2 TOPICAL APPLICATION PRODUCTS IPR-INSTITUTE FOR PHARMACEUTICAL RESEARCH AG (CH) 2000-03-23 WO claimed
US-7910755-B2 Stem cell expansion and uses HARBOR BIOSCIENCES, INC. (US) 2011-03-22 US disclosed
EP-1680076-B1 PHARMACEUTICAL AND COSMETIC FORMULATIONS FOR TREATING FINGERNAILS BIOEQUAL AG (CH) 2008-07-02 EP disclosed
US-20070166249-A1 Pharmaceutical and cosmetic formulations for treating fingernails BIOEQUAL AG (CH) 2007-07-19 US disclosed
US-20070077201-A1 Stem cell expansion and uses BIOVIE INC. 2007-04-05 US disclosed
EP-1680076-A1 PHARMACEUTICAL AND COSMETIC FORMULATIONS FOR TREATING FINGERNAILS BioEqual AG (CH) 2006-07-19 EP disclosed
WO-2005063777-A1 BENZYLPHOSPHATE AND SUBSTITUTED BENZYLPHOSPHATE PRODRUGS FOR THE TREATMENT OF PULMONARY INFLAMMATION CORUS PHARMA (US) 2005-07-14 WO disclosed
EP-1143950-B1 TOPICAL APPLICATION PRODUCTS AGAINST ONYCHOMYCOSES BIOEQUAL AG (CH) 2005-03-09 EP disclosed
WO-2005018585-A1 PHARMACEUTICAL AND COSMETIC FORMULATIONS FOR TREATING FINGERNAILS BIOEQUAL AG (CH) 2005-03-03 WO disclosed
US-6740326-B1 WATER-FREE TOPICAL APPLICATION COMPOSITION FOR TREATMENT OF NAIL DISEASES AND NAIL CARE CONSISTING OF ANTIMYCOTIC AGENT AND LOWER ALKYL ESTER OF LACTIC ACID, MALIC ACID, TARTARIC ACID OR CITRIC ACID AS PENETRATION PROMOTING CARRIER BIOEQUAL AG (CH) 2004-05-25 US disclosed
EP-1143950-A3 TOPICAL APPLICATION PRODUCTS IPR-Institute for Pharmaceutical Research AG (CH) 2002-05-15 EP disclosed
EP-1143950-A2 TOPICAL APPLICATION PRODUCTS IPR-Institute for Pharmaceutical Research AG (CH) 2001-10-17 EP disclosed
WO-2000015202-A2 TOPICAL APPLICATION PRODUCTS IPR-INSTITUTE FOR PHARMACEUTICAL RESEARCH AG (CH) 2000-03-23 WO disclosed
EP-0956047-A1 NEW CARRIER SYSTEMS IPR-Institute for Pharmaceutical Research Riehen AG (CH) 1999-11-17 EP disclosed
WO-1998016251-A1 NEW CARRIER SYSTEMS IPR-INSTITUTE FOR PHARMACEUTICAL RESEARCH AG (CH) 1998-04-23 WO disclosed
EP-0063368-B1 PROCESS FOR THE PREPARATION OF PREGN-4-ENE-3,20-DIONE DERIVATIVES AND 17-ALPHA-ETHYNYL-17-BETA-TRIFLUOROACETOXY-GON-4-ENE-3-ONE DERIVATIVES, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE LATTER COMPOUNDS RICHTER GEDEON VEGYESZETI GYAR R.T. (HU) 1984-07-25 EP disclosed
EP-0063368-A1 Process for the preparation of pregn-4-ene-3,20-dione derivatives and 17-alpha-ethynyl-17-beta-trifluoroacetoxy-gon-4-ene-3-one derivatives, and pharmaceutical compositions containing the latter compounds RICHTER GEDEON VEGYESZETI GYAR R.T. (HU) 1982-10-27 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070077201-A1 Stem cell expansion and uses NES, CD44, FGF2 NR3C1 1099/4885HIF1A 251/4885CYP3A4 4885/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.