Triamcinolone

Triamcinolone

SCHEMBL570639

C[C@]12C=CC(=O)C=C1CC[C@H]1[C@@H]3C[C@@H](O)[C@](O)(C(=O)CO)[C@@]3(C)CC(O)[C@@]12F

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

NR3C1

The experimentally established mechanism targets of Triamcinolone. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR3C1 known ✓ P04150 9/20 1.00
HIF1A Q16665 8/20 1.00
CYP3A4 P08684 7/20 1.00
LMNA P02545 5/20 1.00
HSD17B10 Q99714 4/20 1.00
PGR P06401 4/20 1.00
NFKB1 P19838 3/20 1.00
CYP2C9 P11712 3/20 1.00
PMP22 Q01453 2/20 1.00
CYP2J2 P51589 1/20 1.00
BLM P54132 1/20 1.00
CYP2C19 P33261 1/20 1.00
TSHR P16473 2/20 0.86
AR P10275 2/20 0.86
MEN1 O00255 1/20 0.86
CYP2D6 P10635 1/20 0.86
KMT2A Q03164 1/20 0.86
APEX1 P27695 1/20 0.86
NPSR1 Q6W5P4 1/20 0.86
IKBKB O14920 1/20 0.86

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Triamcinolone SCHEMBL1884154 1.00 NR3C1 (1.00) NR3C1HIF1ACYP3A4LMNAHSD17B10
Triamcinolone SCHEMBL9863653 1.00 NR3C1 (1.00) NR3C1HIF1ACYP3A4LMNAHSD17B10
Triamcinolone SCHEMBL601461 1.00 NR3C1 (1.00) NR3C1HIF1ACYP3A4LMNAHSD17B10
Triamcinolone SCHEMBL1502196 1.00 NR3C1 (1.00) NR3C1HIF1ACYP3A4LMNAHSD17B10
Triamcinolone SCHEMBL14373318 1.00 NR3C1 (1.00) NR3C1HIF1ACYP3A4LMNAHSD17B10
Triamcinolone SCHEMBL8813577 1.00 NR3C1 (1.00) NR3C1HIF1ACYP3A4LMNAHSD17B10
Triamcinolone SCHEMBL24622562 1.00 NR3C1 (1.00) NR3C1HIF1ACYP3A4LMNAHSD17B10
Triamcinolone SCHEMBL601462 1.00 NR3C1 (1.00) NR3C1HIF1ACYP3A4LMNAHSD17B10
Triamcinolone SCHEMBL22962813 1.00 NR3C1 (1.00) NR3C1HIF1ACYP3A4LMNAHSD17B10
Triamcinolone SCHEMBL4447 1.00 NR3C1 (1.00) NR3C1HIF1ACYP3A4LMNAHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 111 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20160206749-A1 METHODS AND COMPOSITIONS FOR ENHANCING DELIVERY OF DOUBLE-STRANDED RNA OR A DOUBLE-STRANDED HYBRID NUCLEIC ACID TO REGULATE GENE EXPRESSION IN MAMMALIAN CELLS MARINA BIOTECH, INC. (US) 2016-07-21 US claimed
US-20080261304-A1 METHODS AND COMPOSITIONS FOR ENHANCING DELIVERY OF DOUBLE-STRANDED RNA OR A DOUBLE-STRANDED HYBRID NUCLEIC ACID TO REGULATE GENE EXPRESSION IN MAMMALIAN CELLS NASTECH PHARMACEUTICAL COMPANY INC. (US) 2008-10-23 US claimed
US-20060014289-A1 Methods and compositions for enhancing delivery of double-stranded RNA or a double-stranded hybrid nucleic acid to regulate gene expression in mammalian cells NASTECH PHARMACEUTICAL COMPANY INC. (US) 2006-01-19 US claimed
US-6830758-B2 Patch containing drug; flexible backing; pressure sensitive adhesive LECTEC CORPORATION 2004-12-14 US claimed
US-20030077316-A1 Psoriasis patch AXOGEN CORPORATION 2003-04-24 US claimed
US-20020192273-A1 Therapeutic patch useful for the treatment of hemorrhoids LEC TEC CORPORATION 2002-12-19 US claimed
EP-0231070-B1 Fluorocarbon blood substitutes ALLIANCE PHARMA (US) 1998-06-10 EP claimed
US-5080885-A Brominated perfluorocarbon emulsions for internal animal use for contrast enhancement and oxygen transport ALLIANCE PHARMACEUTICAL CORP. (US) 1992-01-14 US claimed
EP-0231070-A2 Fluorocarbon blood substitutes ALLIANCE PHARMACEUTICAL CORP. (US) 1987-08-05 EP claimed
US-20230128252-A1 PHARMACEUTICAL COMPOSITIONS Shenzhen Pharmacin Co., Ltd. (CN) 2023-04-27 US disclosed
EP-4135699-A1 PHARMACEUTICAL COMPOSITIONS Shenzhen Pharmacin Co., Ltd. (CN) 2023-02-22 EP disclosed
US-20220135633-A1 METHODS AND SYSTEMS FOR DESIGNING AND/OR CHARACTERIZING SOLUBLE LIPIDATED LIGAND AGENTS ON TARGET THERAPEUTICS LLC 2022-05-05 US disclosed
EP-3692981-B1 TOPICAL COMPOSITION FOR USE IN THE TREATMENT OF PSORIASIS CHEM CURE ASS LLC (US) 2022-05-04 EP disclosed
US-11260063-B2 Method and compositions for treating psoriasis CHEM-CURE ASSOCIATES LLC (US) 2022-03-01 US disclosed
US-4432964-A Topical composition containing steroid in two forms released independently from polymeric carrier ALZA CORPORATION (US) 1984-02-21 US disclosed
US-4304765-A Ocular insert housing steroid in two different therapeutic forms ALZA CORPORATION (US) 1981-12-08 US disclosed
US-4181669-A A CARBODIIMIDE WITH ACID CATALYSTS AS A CONDENSATION AGENT AKTIEBOLAGET LEO (SE) 1980-01-01 US disclosed
US-4180504-A Method for the preparation of esters AKTIEBOLAGET LEO (SE) 1979-12-25 US disclosed
US-4150120-A Ophthalmic TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1979-04-17 US disclosed
US-4112073-A Medicinal composition comprising adrenal cortical hormone and thyroid stimulating hormone releasing hormone TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1978-09-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220135633-A1 METHODS AND SYSTEMS FOR DESIGNING AND/OR CHARACTERIZING SOLUBLE LIPIDATED LIGAND AGENTS LDLR, HDLBP, LIPG NR3C1 3463/4885HIF1A 2861/4885CYP3A4 2859/4885
US-20080261304-A1 METHODS AND COMPOSITIONS FOR ENHANCING DELIVERY OF DOUBLE-STRANDED RNA OR A DOUBLE-STRANDED HYBRID NUCLEIC ACID TO REGULATE GENE EXPRESSION IN MAMMALIAN CELLS SNRPE, LDLR, SNRPA NR3C1 905/4885HIF1A 789/4885CYP3A4 4883/4885
US-20160206749-A1 METHODS AND COMPOSITIONS FOR ENHANCING DELIVERY OF DOUBLE-STRANDED RNA OR A DOUBLE-STRANDED HYBRID NUCLEIC ACID TO REGULATE GENE EXPRESSION IN MAMMALIAN CELLS SNRPE, SREBF2, SREBF1 NR3C1 3285/4885HIF1A 1123/4885CYP3A4 4860/4885
US-20020192273-A1 Therapeutic patch useful for the treatment of hemorrhoids PTGIR, PLOD3, PTGIS NR3C1 2462/4885HIF1A 674/4885CYP3A4 4474/4885
US-20230128252-A1 PHARMACEUTICAL COMPOSITIONS SLCO4C1, SLCO1B1, SLCO1A2 NR3C1 4012/4885HIF1A 3654/4885CYP3A4 38/4885
US-20060014289-A1 Methods and compositions for enhancing delivery of double-stranded RNA or a double-stranded hybrid nucleic acid to regulate gene expression in mammalian cells SNRPE, SREBF2, SREBF1 NR3C1 3285/4885HIF1A 1123/4885CYP3A4 4860/4885
US-20030077316-A1 Psoriasis patch PEF1, ITCH, DSG1 NR3C1 1592/4885HIF1A 1316/4885CYP3A4 4756/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.