SCHEMBL15028344

SCHEMBL15028344

COC(=O)c1sccc1OC1CCN(C(=O)OC(C)(C)C)CC1

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 3/20 0.50
PDE4D Q08499 3/20 0.50
PDE4A P27815 2/20 0.50
PDE4C Q08493 2/20 0.50
GPR119 Q8TDV5 7/20 0.49
ALDH1A1 P00352 2/20 0.48
KDM1A O60341 1/20 0.47
EED O75530 1/20 0.47
RBBP4 Q09028 1/20 0.47
SUZ12 Q15022 1/20 0.47
EZH2 Q15910 1/20 0.47
AEBP2 Q6ZN18 1/20 0.47
PTPN2 P17706 1/20 0.45
PTPN1 P18031 1/20 0.45
PTPN6 P29350 1/20 0.45
STS P08842 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15028316 0.88 PDE4B (0.49) PDE4BPDE4DPDE4APDE4CGPR119
SCHEMBL7486842 0.82 ALDH1A1 (0.60) ALDH1A1EEDRBBP4SUZ12EZH2
SCHEMBL2424923 0.81 ALDH1A1 (0.50) GPR119ALDH1A1EEDRBBP4SUZ12
SCHEMBL31078515 0.80 PDE4B (0.48) PDE4BPDE4DPDE4APDE4CGPR119
SCHEMBL31078714 0.80 PDE4B (0.48) PDE4BPDE4DPDE4APDE4CGPR119
SCHEMBL16296065 0.79 KDM1A (0.53) PDE4BPDE4DPDE4APDE4CGPR119
SCHEMBL3158355 0.78 PDE4B (0.49) PDE4BPDE4DPDE4APDE4CGPR119
SCHEMBL13060447 0.78 PDE4D (0.49) PDE4BPDE4DPDE4APDE4CGPR119
SCHEMBL3898794 0.78 ALDH1A1 (0.46) PDE4BALDH1A1
SCHEMBL3151620 0.78 STS (0.55) PDE4BPDE4DPDE4APDE4CGPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013083991-A1 NOVEL COMPOUNDS AND THEIR USE IN THERAPY IMPERIAL INNOVATIONS LIMITED (GB) 2013-06-13 WO disclosed