SCHEMBL1503299

SCHEMBL1503299

COC(=O)c1ncc(COc2ccc(F)cc2)c(CONC(=O)c2ncc(COc3ccc(F)c(Cl)c3)c(CO)c2O)c1O

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 5/20 0.36
SCN5A Q14524 1/20 0.34
ADAMTS4 O75173 1/20 0.34
MMP2 P08253 1/20 0.34
MMP13 P45452 1/20 0.34
MMP14 P50281 1/20 0.34
ADAMTS5 Q9UNA0 1/20 0.34
ALDH1A1 P00352 3/20 0.33
GSTP1 P09211 1/20 0.33
PARP14 Q460N5 1/20 0.33
PARP10 Q53GL7 1/20 0.33
KMT2A Q03164 3/20 0.33
MEN1 O00255 2/20 0.33
GAA P10253 1/20 0.32
KLKB1 P03952 1/20 0.32
POLB P06746 1/20 0.32
LMNA P02545 1/20 0.32
MAPT P10636 1/20 0.32
HPGD P15428 1/20 0.32
MAOB P27338 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1503300 0.92 ADAMTS4 (0.37) SCN9ASCN5AADAMTS4MMP2MMP13
SCHEMBL2220322 0.89 ALDH1A1 (0.40) SCN9ASCN5AALDH1A1KMT2AMEN1
SCHEMBL1503187 0.83 ALDH1A1 (0.41) ALDH1A1PARP10KMT2AMEN1GAA
SCHEMBL22738223 0.82 SCN9A (0.41) SCN9ASCN5AMAPTMAOBMAOA
SCHEMBL30954808 0.82 HDAC1 (0.41) SCN9ASCN5AMAPTMAOB
SCHEMBL1503267 0.82 HDAC1 (0.41) SCN9ASCN5AMAPTMAOB
SCHEMBL22719903 0.80 GRIN1 (0.43) SCN9ASCN5AALDH1A1KLKB1LMNA
SCHEMBL22738285 0.79 MEN1 (0.40) SCN9ASCN5AKMT2AMEN1KLKB1
SCHEMBL4304503 0.78 PPARG (0.41) SCN9ASCN5AMAPTMAOBMAOA
SCHEMBL1503165 0.77 ALDH1A1 (0.41) SCN9ASCN5AALDH1A1KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2300433-A1 HIV INTEGRASE INHIBITORS FROM PYRIDOXINE Ambrilia Biopharma Inc. (CA) 2011-03-30 EP disclosed
WO-2009146555-A1 HIV INTEGRASE INHIBITORS FROM PYRIDOXINE AMBRILIA BIOPHARMA INC. (CA) 2009-12-10 WO disclosed