SCHEMBL15033256

SCHEMBL15033256

CNC(=O)[C@@H](NC(=O)[C@@H](NC)C(C)C)C(C)C

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MMP1 P03956 1/20 0.38
MMP9 P14780 1/20 0.38
MMP14 P50281 1/20 0.38
FFAR2 O15552 1/20 0.32
POLB P06746 1/20 0.32
CNR2 P34972 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.31
CTSS P25774 1/20 0.31
CTSK P43235 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22421642 1.00 MMP1 (0.38) MMP1MMP9MMP14FFAR2POLB
SCHEMBL29878045 1.00 MMP1 (0.38) MMP1MMP9MMP14FFAR2POLB
SCHEMBL24337164 1.00 MMP1 (0.38) MMP1MMP9MMP14FFAR2POLB
SCHEMBL19401641 0.91 FFAR2 (0.36) MMP1MMP9MMP14FFAR2
SCHEMBL13260893 0.91 FFAR2 (0.36) MMP1MMP9MMP14FFAR2
SCHEMBL14511336 0.91 FFAR2 (0.36) MMP1MMP9MMP14FFAR2
SCHEMBL17305511 0.84 SMN1; SMN2 (0.42) POLBSMN1; SMN2
SCHEMBL19201191 0.84 FFAR2 (0.32) MMP1FFAR2
SCHEMBL19201193 0.84 FFAR2 (0.32) MMP1FFAR2
SCHEMBL26789813 0.84 MMP1 (0.38) MMP1MMP9MMP14FFAR2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240216526-A1 PREPARATION METHOD FOR DUAL-DRUG-LINKER OF ADC AND USE THEREOF CHENGDU SCIMOUNT PHARMATECH CO., LTD. (CN) 2024-07-04 US disclosed
WO-2024052333-A1 MULTIVALENT FIBROBLAST ACTIVATION PROTEIN LIGANDS FOR TARGETED DELIVERY APPLICATIONS PHILOCHEM AG (CH) 2024-03-14 WO disclosed
WO-2023144379-A1 HIGH-AFFINITY LIGANDS OF FIBROBLAST ACTIVATION PROTEIN FOR TARGETED DELIVERY APPLICATIONS PHILOCHEM AG (CH) 2023-08-03 WO disclosed
WO-2021129678-A1 CONJUGATE WITH RADIATION-RESPONSIVE GROUP AND USE THEREOF 北京大学 2021-07-01 WO disclosed
EP-2898085-B1 CELL LINES MEDIMMUNE LTD (GB) 2019-01-23 EP disclosed
EP-3327027-A1 CYTOTOXIC PEPTIDES AND ANTIBODY DRUG CONJUGATES THEREOF Pfizer Inc (US) 2018-05-30 EP disclosed
EP-3284751-A1 ANTI-C-MET ANTIBODY AND ANTI-C-MET ANTIBODY-CYTOTOXIC DRUG CONJUGATE AND PHARMACEUTICAL USE THEREOF Suzhou Suncadia Biopharmaceuticals Co., Ltd. (CN) 2018-02-21 EP disclosed
US-9217015-B2 Cyclosporin derivatives for the treatment and prevention of a viral infection S&T GLOBAL INC. (US) 2015-12-22 US disclosed
US-20130303438-A1 NOVEL CYCLOSPORIN DERIVATIVES FOR THE TREATMENT AND PREVENTION OF A VIRAL INFECTION S&T GLOBAL INC. 2013-11-14 US disclosed
WO-2013085925-A1 ANTIBODY-DRUG CONJUGATES AND RELATED COMPOUNDS, COMPOSITIONS, AND METHODS IGENICA, INC. (US) 2013-06-13 WO disclosed
WO-2012166560-A1 COMPOSITIONS CONTAINING, METHODS INVOLVING, AND USES OF NON-NATURAL AMINO ACID LINKED DOLASTATIN DERIVATIVES AMBRX, INC. (US) 2012-12-06 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130303438-A1 NOVEL CYCLOSPORIN DERIVATIVES FOR THE TREATMENT AND PREVENTION OF A VIRAL INFECTION HAVCR2, TSLP, ICOS MMP1 3789/4885MMP9 4062/4885MMP14 2421/4885
US-20240216526-A1 PREPARATION METHOD FOR DUAL-DRUG-LINKER OF ADC AND USE THEREOF SKP1, ADCY7, ERBB2 MMP1 4315/4885MMP9 3233/4885MMP14 3717/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.