SCHEMBL15041024

SCHEMBL15041024

CCn1ncc2c(oc3c(OC(F)F)ccc(C)c32)c1=O

nearest known ligand 0.32

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 6/20 0.32
NPC1 O15118 1/20 0.32
CRHR1 P34998 1/20 0.32
PDE1A P54750 1/20 0.31
PDE1B Q01064 1/20 0.31
PDE1C Q14123 1/20 0.31
PDE4D Q08499 3/20 0.31
PDE4A P27815 2/20 0.31
PDE4B Q07343 2/20 0.31
PDE4C Q08493 2/20 0.31
GRIN1 Q05586 3/20 0.31
GRIN2B Q13224 3/20 0.31
CYP17A1 P05093 1/20 0.30
CYP19A1 P11511 1/20 0.30
CYP11B1 P15538 1/20 0.30
CYP11B2 P19099 1/20 0.30
TRPA1 O75762 1/20 0.30
CTSD P07339 1/20 0.30
BACE2 Q9Y5Z0 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL73417 0.85 PDE4D (0.38) NPC1PDE4DPDE4APDE4BPDE4C
SCHEMBL73992 0.85 PDE4B (0.39) NPC1PDE4DPDE4APDE4BPDE4C
SCHEMBL73786 0.77 PDE4D (0.57) PDE4DPDE4APDE4BPDE4C
SCHEMBL73917 0.76 PDE4D (0.36) PDE4DPDE4APDE4BPDE4C
SCHEMBL73069 0.76 MAPT (0.40) PDE4DPDE4APDE4BPDE4C
SCHEMBL5504865 0.76 ALDH1A1 (0.39) PDE4DPDE4APDE4BPDE4C
SCHEMBL26906599 0.71 GAA (0.37) CRHR1PDE1APDE1BPDE1CGRIN1
SCHEMBL75082 0.71 ALDH1A1 (0.44) NPC1PDE4DPDE4APDE4BPDE4C
SCHEMBL85521 0.69 PDE4D (0.54) PDE4DPDE4APDE4BPDE4C
SCHEMBL3873741 0.69 PDE4B (0.36) PDE4DPDE4APDE4BPDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1831227-B1 NOVEL HETEROCYCLIC COMPOUNDS USEFUL FOR THE TREATMENT OF INFLAMMATORY AND ALLERGIC DISORDERS GLENMARK PHARMACEUTICALS SA (CH) 2013-06-19 EP disclosed