SCHEMBL15042495

SCHEMBL15042495

O=[PH](O)OCCCNCc1cc(-c2ccco2)c(OCCCCCc2ccccc2)cc1F

nearest known ligand 0.37

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.36
S1PR1 P21453 2/20 0.34
S1PR3 Q99500 1/20 0.34
S1PR5 Q9H228 1/20 0.34
FAAH O00519 1/20 0.34
CES1 P23141 1/20 0.34
KDM4E B2RXH2 3/20 0.33
SIGMAR1 Q99720 2/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
CNR1 P21554 1/20 0.33
CNR2 P34972 1/20 0.33
BCHE P06276 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15042579 0.94 ALDH1A1 (0.34) ALDH1A1S1PR1S1PR3KDM4EKMT2A
SCHEMBL15042635 0.92 MPO (0.38) ALDH1A1MEN1KMT2A
SCHEMBL15042607 0.86 ALDH1A1 (0.39) ALDH1A1S1PR1S1PR3S1PR5KDM4E
SCHEMBL15022603 0.86 S1PR2 (0.47) S1PR1S1PR3S1PR5
SCHEMBL15042598 0.85 SLC6A5 (0.35) ALDH1A1KDM4EKMT2A
SCHEMBL15042476 0.83 S1PR2 (0.37) ALDH1A1S1PR1S1PR3KDM4EMEN1
SCHEMBL15042584 0.83 MPO (0.40) ALDH1A1MEN1KMT2A
SCHEMBL15042532 0.83 KMT2A (0.39) ALDH1A1S1PR1S1PR3KDM4EMEN1
SCHEMBL15042553 0.82 ALDH1A1 (0.36) ALDH1A1S1PR1S1PR3KDM4EMEN1
SCHEMBL15042494 0.82 SLC6A5 (0.35) KDM4EKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8828973-B2 Compounds as receptor modulators with therapeutic utility ALLERGAN, INC. (US) 2014-09-09 US disclosed
US-20140221317-A1 NOVEL COMPOUNDS AS RECEPTOR MODULATORS WITH THERAPEUTIC UTILITY ALLERGAN, INC. (US) 2014-08-07 US disclosed
US-8741875-B2 Compounds as receptor modulators with therapeutic utility ALLERGAN, INC. (US) 2014-06-03 US disclosed
US-20130157982-A1 NOVEL COMPOUNDS AS RECEPTOR MODULATORS WITH THERAPEUTIC UTILITY ALLERGAN, INC. (US) 2013-06-20 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140221317-A1 NOVEL COMPOUNDS AS RECEPTOR MODULATORS WITH THERAPEUTIC UTILITY S1PR1, S1PR3, S1PR2 ALDH1A1 3552/4885S1PR1 1/4885S1PR3 2/4885
US-20130157982-A1 NOVEL COMPOUNDS AS RECEPTOR MODULATORS WITH THERAPEUTIC UTILITY S1PR1, S1PR3, S1PR2 ALDH1A1 3552/4885S1PR1 1/4885S1PR3 2/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.