SCHEMBL15045205

SCHEMBL15045205

C[C@H](N)C(=O)N(C)C1CCN(C)CC1

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.43
CCR5 P51681 2/20 0.42
ALDH1A1 P00352 2/20 0.40
LMNA P02545 2/20 0.40
KDM4E B2RXH2 2/20 0.38
KMT2A Q03164 1/20 0.37
HTR2A P28223 1/20 0.37
HTR2C P28335 1/20 0.37
POLB P06746 1/20 0.36
BRD4 O60885 1/20 0.36
TAF1 P21675 1/20 0.36
CECR2 Q9BXF3 1/20 0.36
DPP4 P27487 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19502748 1.00 HTT (0.43) HTTCCR5ALDH1A1LMNAKDM4E
SCHEMBL800697 0.85 HTT (0.45) HTTCCR5ALDH1A1LMNAKDM4E
SCHEMBL19882800 0.81 ALDH1A1 (0.40) CCR5ALDH1A1DPP4
SCHEMBL5498956 0.79 FAAH (0.42) ALDH1A1
SCHEMBL12022268 0.77 ALDH1A1 (0.48) ALDH1A1LMNAKDM4EKMT2AHTR2A
SCHEMBL7979611 0.77 ALDH1A1 (0.48) ALDH1A1LMNAKDM4EKMT2AHTR2A
SCHEMBL8191420 0.77 HTT (0.43) HTTCCR5ALDH1A1LMNAKDM4E
SCHEMBL14155233 0.77 HTT (0.43) HTTCCR5ALDH1A1LMNAKDM4E
SCHEMBL15029872 0.77 GAA (0.51) HTTALDH1A1LMNAKDM4EKMT2A
SCHEMBL13808539 0.76 HTT (0.42) HTTCCR5ALDH1A1LMNAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3464273-B9 IMIDAZOLONE COMPOUNDS AS HUMAN NEUTROPHIL ELASTASE INHIBITORS CHIESI FARM SPA (IT) 2020-10-21 EP disclosed
EP-3464273-B1 IMIDAZOLONE COMPOUNDS AS HUMAN NEUTROPHIL ELASTASE INHIBITORS CHIESI FARM SPA (IT) 2020-04-08 EP disclosed
EP-3464268-B1 NOVEL COMPOUNDS CHIESI FARM SPA (IT) 2020-03-11 EP disclosed
EP-2604601-A1 HETERO RING COMPOUND Astellas Pharma Inc. (JP) 2013-06-19 EP disclosed