SCHEMBL15045453

SCHEMBL15045453

Cc1cc2c([nH]1)Cc1ccccc1CC2

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.41
DRD1 P21728 13/20 0.40
DRD2 P14416 12/20 0.40
DRD5 P21918 12/20 0.40
DRD3 P35462 9/20 0.40
DRD4 P21917 9/20 0.40
KDM4E B2RXH2 1/20 0.40
MEN1 O00255 1/20 0.40
GMNN O75496 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
ADRA1D P25100 1/20 0.40
CYP2C19 P33261 1/20 0.40
ADRA1A P35348 1/20 0.40
ADRA1B P35368 1/20 0.40
MTOR P42345 1/20 0.40
BLM P54132 1/20 0.40
PMP22 Q01453 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15045572 0.87 DRD1 (0.42) CYP2A6DRD1DRD2DRD5DRD3
SCHEMBL15042875 0.77 DRD5 (0.43) CYP2A6DRD1DRD2DRD5DRD3
SCHEMBL19229361 0.73 ALDH1A1 (0.40) KDM4ECYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL15045569 0.73 TYMS (0.51) CYP2A6DRD1DRD2DRD5DRD3
SCHEMBL15045455 0.70 PARP1 (0.35) DRD1DRD2DRD5DRD3DRD4
SCHEMBL7959781 0.69 ALDH1A1 (0.46) KDM4EMEN1KMT2ATSHRALOX15
SCHEMBL12844664 0.69
SCHEMBL250734 0.68 CYP2A6 (0.65) CYP2A6DRD1DRD2DRD5DRD3
SCHEMBL13029239 0.68 PNMT (0.40) DRD2DRD3PNMTCD44MAOB
SCHEMBL19485911 0.68 HTR2A (0.37) KDM4EMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9796705-B2 Fused tricyclic compounds and methods of use thereof for the treatment of viral diseases MERCK SHARP & DOHME CORP. (US) 2017-10-24 US disclosed
US-20130156731-A1 FUSED TRICYCLIC COMPOUNDS AND METHODS OF USE THEREOF FOR THE TREATMENT OF VIRAL DISEAS SCHERING CORPORATION 2013-06-20 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130156731-A1 FUSED TRICYCLIC COMPOUNDS AND METHODS OF USE THEREOF FOR THE TREATMENT OF VIRAL DISEAS HAVCR2, ELOC, ZC3HAV1 CYP2A6 256/4885DRD1 2549/4885DRD2 2849/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.