SCHEMBL15055063

SCHEMBL15055063

C#CCC(Cc1cnc2nc(N)nc(O)c2n1)(C(=O)O)c1ccc(C(=O)O)cc1

nearest known ligand 0.38

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
DHFR P00374 14/20 0.38
FOLR1 P15328 1/20 0.38
SLC19A1 P41440 1/20 0.38
SLC46A1 Q96NT5 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15054326 0.92 DHFR (0.46) DHFRFOLR1SLC19A1SLC46A1
SCHEMBL17562254 0.77 DHFR (0.46) DHFRFOLR1SLC19A1SLC46A1
SCHEMBL17554357 0.77 DHFR (0.46) DHFRFOLR1SLC19A1SLC46A1
SCHEMBL17554406 0.77 DHFR (0.46) DHFRFOLR1SLC19A1SLC46A1
SCHEMBL17554417 0.77 DHFR (0.46) DHFRFOLR1SLC19A1SLC46A1
Pteroic Acid SCHEMBL245982 0.71 DHFR (0.67) DHFR
SCHEMBL17554416 0.71 DHFR (0.44) DHFRFOLR1SLC19A1SLC46A1
Potassium Ion SCHEMBL17554403 0.71 DHFR (0.44) DHFRFOLR1SLC19A1SLC46A1
SCHEMBL15055069 0.71 NOS1 (0.35) DHFR
Pteroic Acid SCHEMBL16047869 0.70 DHFR (0.66) DHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2794610-B1 PROCESSES AND INTERMEDIATES FOR PREPARING PRALATREXATE PLUS CHEMICALS SA (CH) 2016-03-09 EP disclosed
EP-2794610-A1 PROCESSES AND INTERMEDIATES FOR PREPARING PRALATREXATE Plus Chemicals SA (CH) 2014-10-29 EP disclosed
WO-2013096800-A1 PROCESSES AND INTERMEDIATES FOR PREPARING PRALATREXATE PLUS CHEMICALS S.A. (CH) 2013-06-27 WO disclosed