SCHEMBL15062809

SCHEMBL15062809

COc1cc(C)c(S(=O)(=O)N2CCc3ccc(OC(=O)O)cc3C2)c(C)c1

nearest known ligand 0.58

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 10/20 0.58
PKM P14618 2/20 0.49
CYP3A4 P08684 1/20 0.43
CYP2C19 P33261 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
LMNA P02545 1/20 0.43
RAB9A P51151 1/20 0.42
PDE4B Q07343 1/20 0.42
PDE4D Q08499 1/20 0.42
PPARG P37231 1/20 0.41
PPARD Q03181 1/20 0.41
PPARA Q07869 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
AKR1C1 Q04828 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15062737 0.91 AKR1C3 (0.46) AKR1C3PKMSMN1; SMN2L3MBTL1AKR1C1
SCHEMBL3100375 0.87 AKR1C3 (0.64) AKR1C3PKMAKR1C1
SCHEMBL3091050 0.84 AKR1C3 (0.50) AKR1C3PKMCYP3A4CYP2C19SMN1; SMN2
SCHEMBL3079208 0.83 AKR1C3 (0.52) AKR1C3PKMSMN1; SMN2LMNARAB9A
SCHEMBL3722871 0.83 PKM (0.49) AKR1C3PKMCYP3A4CYP2C19SMN1; SMN2
SCHEMBL3091835 0.82 AKR1C3 (0.47) AKR1C3PKMCYP3A4CYP2C19SMN1; SMN2
SCHEMBL15062765 0.82 MEN1 (0.49) AKR1C3SMN1; SMN2LMNAPDE4BPDE4D
SCHEMBL15062792 0.78 L3MBTL1 (0.51) AKR1C3L3MBTL1MEN1KMT2A
SCHEMBL15062805 0.78 AKR1C3 (0.43) AKR1C3MEN1KMT2A
SCHEMBL3088744 0.78 PKM (0.44) AKR1C3PKMCYP3A4CYP2C19SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2393812-B1 SUBSTITUTED SPIROAMIDES AS B1R-MODULATORS GRUENENTHAL GMBH (DE) 2013-07-03 EP disclosed