SCHEMBL15062890

SCHEMBL15062890

CC(=O)CNC[C@H](O)[C@@H](Cc1cc(F)ccc1F)NC(=O)OC(C)(C)C

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 2/20 0.40
BACE1 P56817 4/20 0.40
KLK5 Q9Y337 2/20 0.40
GPR119 Q8TDV5 1/20 0.40
CTSS P25774 3/20 0.38
CTSK P43235 3/20 0.38
CTSD P07339 2/20 0.37
PTPN1 P18031 1/20 0.36
ATM Q13315 1/20 0.36
DPP4 P27487 2/20 0.34
DPP7 Q9UHL4 2/20 0.34
DPP8 Q6V1X1 1/20 0.34
DPP9 Q86TI2 1/20 0.34
RIPK1 Q13546 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL496196 0.87 SCN9A (0.42) SCN9ABACE1KLK5GPR119CTSS
SCHEMBL496197 0.87 SCN9A (0.42) SCN9ABACE1KLK5GPR119CTSS
SCHEMBL495863 0.84 KLK5 (0.43) SCN9AKLK5GPR119CTSSCTSK
SCHEMBL495865 0.84 KLK5 (0.43) SCN9AKLK5GPR119CTSSCTSK
SCHEMBL496081 0.82 RIPK1 (0.41) SCN9AKLK5GPR119CTSSCTSK
SCHEMBL496083 0.82 RIPK1 (0.41) SCN9AKLK5GPR119CTSSCTSK
SCHEMBL15062933 0.78 KLK5 (0.59) BACE1KLK5CTSSCTSKATM
SCHEMBL10074464 0.77 SCN9A (0.49) SCN9AGPR119CTSSCTSKPTPN1
SCHEMBL6873438 0.76 CTSK (0.47) SCN9AGPR119CTSSCTSKPTPN1
SCHEMBL269147 0.75 SCN9A (0.45) SCN9AKLK5CTSSCTSKPTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1910317-B1 1-AMINO LINKED COMPOUNDS LILLY CO ELI (US) 2013-07-03 EP disclosed