SCHEMBL15062986

SCHEMBL15062986

CC#CC(NCC(CSCC1CC1)C(=O)NC1(C#N)CC1)C(F)(F)Oc1ccc(SC)cc1

nearest known ligand 0.36

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CTSL P07711 13/20 0.36
CTSK P43235 5/20 0.36
CTSS P25774 4/20 0.36
CTSB P07858 3/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15062985 1.00 CTSL (0.36) CTSLCTSKCTSSCTSB
SCHEMBL15062901 0.89 CTSL (0.43) CTSLCTSKCTSSCTSB
SCHEMBL15062902 0.89 CTSL (0.43) CTSLCTSKCTSSCTSB
SCHEMBL15062930 0.83 CTSL (0.38) CTSLCTSKCTSSCTSB
SCHEMBL15062929 0.83 CTSL (0.38) CTSLCTSKCTSSCTSB
SCHEMBL15062778 0.79 LNPEP (0.31)
SCHEMBL15062780 0.79 LNPEP (0.31)
SCHEMBL15062943 0.78 ACE (0.35) CTSLCTSKCTSSCTSB
SCHEMBL15062942 0.78 ACE (0.35) CTSLCTSKCTSSCTSB
SCHEMBL2401476 0.77 CTSL (0.53) CTSLCTSKCTSSCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2361243-B9 HALOALKYL CONTAINING COMPOUNDS AS CYSTEINE PROTEASE INHIBITORS VIROBAY INC (US) 2014-06-11 EP disclosed
EP-2361243-B1 HALOALKYL CONTAINING COMPOUNDS AS CYSTEINE PROTEASE INHIBITORS VIROBAY INC (US) 2013-07-03 EP disclosed