SCHEMBL15066568

SCHEMBL15066568

O=C(O)NCC(O)Cc1ccc(Cl)cc1Cl

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 8/20 0.45
ALDH1A1 P00352 2/20 0.45
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
HPGD P15428 1/20 0.44
CNR1 P21554 1/20 0.43
CYP3A4 P08684 2/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2D6 P10635 1/20 0.42
ALOX15 P16050 1/20 0.42
CYP2C19 P33261 1/20 0.42
GGPS1 O95749 1/20 0.42
METAP2 P50579 1/20 0.42
CYP2C9 P11712 1/20 0.41
HDAC3 O15379 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC2 Q92769 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16054409 0.85 METAP2 (0.48) ALDH1A1MEN1KMT2AHPGDCNR1
SCHEMBL5433210 0.84 OPRK1 (0.51) HDAC8ALDH1A1MEN1KMT2ACNR1
SCHEMBL248588 0.83 HDAC8 (0.46) HDAC8ALDH1A1MEN1KMT2ACYP3A4
SCHEMBL19254238 0.83 HDAC8 (0.46) HDAC8ALDH1A1MEN1KMT2AHPGD
SCHEMBL5436525 0.82 KMT2A (0.63) ALDH1A1MEN1KMT2AHPGDCNR1
SCHEMBL19254537 0.81 NPC1 (0.49) ALDH1A1MEN1KMT2A
SCHEMBL15067896 0.81 NPC1 (0.49) ALDH1A1MEN1KMT2A
SCHEMBL13941148 0.77 IDO1 (0.47) HDAC8CYP3A4CYP1A2CYP2C19GGPS1
SCHEMBL697972 0.77 ALDH1A1 (0.63) ALDH1A1CNR1GGPS1
SCHEMBL8591917 0.77 IDO1 (0.47) HDAC8CYP3A4CYP1A2CYP2C19GGPS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 20 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2970112-A1 PHENYL CARBAMATE COMPOUND AND A COMPOSITION FOR PREVENTING OR TREATING A MEMORY LOSS-RELATED DISEASE COMPRISING THE SAME Bio-Pharm Solutions Co., Ltd. (KR) 2016-01-20 EP claimed
EP-2970111-A1 PHENYL CARBAMATE COMPOUND AND A COMPOSITION FOR PREVENTING OR TREATING A NERVE GAS-INDUCED DISEASE COMPRISING THE SAME Bio-Pharm Solutions Co., Ltd. (KR) 2016-01-20 EP claimed
EP-2970109-A1 PHENYL CARBAMATE COMPOUND AND A COMPOSITION FOR NEUROPROTECTION COMPRISING THE SAME Bio-Pharm Solutions Co., Ltd. (KR) 2016-01-20 EP claimed
EP-2970110-A1 PHENYL CARBAMATE COMPOUND AND A COMPOSITION FOR PREVENTING OR TREATING A PSYCHIATRIC DISORDER COMPRISING THE SAME Bio-Pharm Solutions Co., Ltd. (KR) 2016-01-20 EP claimed
WO-2014142549-A1 PHENYL CARBAMATE COMPOUND AND A COMPOSITION FOR PREVENTING OR TREATING A MEMORY LOSS-RELATED DISEASE COMPRISING THE SAME BIO-PHARM SOLUTIONS CO., LTD. (KR) 2014-09-18 WO claimed
WO-2014142548-A1 PHENYL CARBAMATE COMPOUND AND A COMPOSITION FOR PREVENTING OR TREATING A NERVE GAS-INDUCED DISEASE COMPRISING THE SAME BIO-PHARM SOLUTIONS CO., LTD. (KR) 2014-09-18 WO claimed
WO-2014142547-A1 PHENYL CARBAMATE COMPOUND AND A COMPOSITION FOR NEUROPROTECTION COMPRISING THE SAME BIO-PHARM SOLUTIONS CO., LTD. (KR) 2014-09-18 WO claimed
WO-2014142550-A1 PHENYL CARBAMATE COMPOUND AND A COMPOSITION FOR PREVENTING OR TREATING A PSYCHIATRIC DISORDER COMPRISING THE SAME BIO-PHARM SOLUTIONS CO., LTD. (KR) 2014-09-18 WO claimed
EP-2970112-A1 PHENYL CARBAMATE COMPOUND AND A COMPOSITION FOR PREVENTING OR TREATING A MEMORY LOSS-RELATED DISEASE COMPRISING THE SAME Bio-Pharm Solutions Co., Ltd. (KR) 2016-01-20 EP disclosed
EP-2970111-A1 PHENYL CARBAMATE COMPOUND AND A COMPOSITION FOR PREVENTING OR TREATING A NERVE GAS-INDUCED DISEASE COMPRISING THE SAME Bio-Pharm Solutions Co., Ltd. (KR) 2016-01-20 EP disclosed
EP-2970109-A1 PHENYL CARBAMATE COMPOUND AND A COMPOSITION FOR NEUROPROTECTION COMPRISING THE SAME Bio-Pharm Solutions Co., Ltd. (KR) 2016-01-20 EP disclosed
EP-2970110-A1 PHENYL CARBAMATE COMPOUND AND A COMPOSITION FOR PREVENTING OR TREATING A PSYCHIATRIC DISORDER COMPRISING THE SAME Bio-Pharm Solutions Co., Ltd. (KR) 2016-01-20 EP disclosed
EP-2968211-A1 PHENYL ALKYL CARBAMATE COMPOUNDS FOR USE IN PREVENTING OR TREATING EPILEPSY OR EPILEPSY-RELATED SYNDROME Bio-Pharm Solutions Co., Ltd. (KR) 2016-01-20 EP disclosed
EP-2797881-A1 Phenyl alkyl carbamate derivative compound and pharmaceutical composition containing the same Bio-Pharm Solutions Co., Ltd. (KR) 2014-11-05 EP disclosed
WO-2014142549-A1 PHENYL CARBAMATE COMPOUND AND A COMPOSITION FOR PREVENTING OR TREATING A MEMORY LOSS-RELATED DISEASE COMPRISING THE SAME BIO-PHARM SOLUTIONS CO., LTD. (KR) 2014-09-18 WO disclosed
WO-2014142548-A1 PHENYL CARBAMATE COMPOUND AND A COMPOSITION FOR PREVENTING OR TREATING A NERVE GAS-INDUCED DISEASE COMPRISING THE SAME BIO-PHARM SOLUTIONS CO., LTD. (KR) 2014-09-18 WO disclosed
WO-2014142547-A1 PHENYL CARBAMATE COMPOUND AND A COMPOSITION FOR NEUROPROTECTION COMPRISING THE SAME BIO-PHARM SOLUTIONS CO., LTD. (KR) 2014-09-18 WO disclosed
WO-2014142550-A1 PHENYL CARBAMATE COMPOUND AND A COMPOSITION FOR PREVENTING OR TREATING A PSYCHIATRIC DISORDER COMPRISING THE SAME BIO-PHARM SOLUTIONS CO., LTD. (KR) 2014-09-18 WO disclosed
WO-2014142519-A1 PHENYL ALKYL CARBAMATE COMPOUNDS FOR USE IN PREVENTING OR TREATING EPILEPSY OR EPILEPSY-RELATED SYNDROME BIO-PHARM SOLUTIONS CO., LTD. (KR) 2014-09-18 WO disclosed
WO-2013100566-A1 Phenyl alkyl carbamate derivative compound and pharmaceutical composition containing the same BIO-PHARM SOLUTIONS CO., LTD. (KR) 2013-07-04 WO disclosed