Amorolfine

Amorolfine

SCHEMBL150666

CCC(C)(C)c1ccc(CC(C)CN2C[C@@H](C)O[C@@H](C)C2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 1/20 1.00
CHRM1 P11229 1/20 1.00
DRD3 P35462 1/20 1.00
KCNH2 Q12809 1/20 1.00
SIGMAR1 Q99720 3/20 0.79
EBP Q15125 1/20 0.79
HRH3 Q9Y5N1 12/20 0.40
MAOB P27338 4/20 0.40
MAPK1 P28482 1/20 0.39
L3MBTL1 Q9Y468 2/20 0.38
ALDH1A1 P00352 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Amorolfine SCHEMBL8165433 1.00 ADORA3 (1.00) ADORA3CHRM1DRD3KCNH2SIGMAR1
Amorolfine SCHEMBL933541 1.00 ADORA3 (1.00) ADORA3CHRM1DRD3KCNH2SIGMAR1
Amorolfine SCHEMBL5579008 0.99 ADORA3 (0.97) ADORA3CHRM1DRD3KCNH2SIGMAR1
Amorolfine SCHEMBL36711 0.99 ADORA3 (0.97) ADORA3CHRM1DRD3KCNH2SIGMAR1
Amorolfine SCHEMBL1934866 0.99 ADORA3 (0.97) ADORA3CHRM1DRD3KCNH2SIGMAR1
Amorolfine SCHEMBL1649004 0.97 ADORA3 (0.95) ADORA3CHRM1DRD3KCNH2SIGMAR1
Amorolfine SCHEMBL3820874 0.95 ADORA3 (0.91) ADORA3CHRM1DRD3KCNH2SIGMAR1
Amorolfine SCHEMBL23111397 0.90 ADORA3 (0.81) ADORA3CHRM1DRD3KCNH2SIGMAR1
SCHEMBL19823129 0.90 ADORA3 (0.81) ADORA3CHRM1DRD3KCNH2SIGMAR1
SCHEMBL11164667 0.89 ADORA3 (0.80) ADORA3CHRM1DRD3KCNH2SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 8783 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2026106952-A1 METHODS FOR TREATING CONGENITAL DISORDERS OF GLYCOSYLATION CDG CARE (US) 2026-05-21 WO claimed
EP-4255391-B1 LUMINOL FOR USE IN THE TREATMENT OF SEQUELAE OF A SARS-COV-2 INFECTION METRIOPHARM AG (CH) 2026-05-06 EP claimed
US-20260102419-A1 USE OF COMPOUNDS IN THE TREATMENT OF FUNGAL INFECTIONS BASILEA PHARMACEUTICA INTERNATIONAL AG, ALLSCHWIL (CH) 2026-04-16 US claimed
EP-4719384-A2 COMPOUNDS WITH ANTIFUNGAL PROPERTIES Trustees of Dartmouth College (US) 2026-04-08 EP claimed
US-20260076924-A1 COMPOSITIONS AND METHODS OF TREATMENT FOR TINEA PEDIS THERAPEUTICS INC (US) 2026-03-19 US claimed
US-20260027255-A1 Cross-Linked Telechelic Polymer Compositions, Methods of Preparation Thereof, and Methods of Using Same BETTY YU SKIN TECH ADVISORS LLC (US) 2026-01-29 US claimed
EP-4680240-A1 METHOD OF TREATING DISORDERS WITH SURF1 MALFUNCTION Cure Mito Foundation (US) 2026-01-21 EP claimed
US-20260007753-A1 DERMAL SKIN PROTECTANT AND CARRIER INSPIRED MAT STRATEGIES LLC (US) 2026-01-08 US claimed
US-20250319078-A1 METHOD FOR SYNERGISTIC ENHANCEMENT OF REMYELINATION VIA MODULATION OF RXR AND A HETERODIMERIC PARTNER LAIRSON LUKE L (US) 2025-10-16 US claimed
US-12433856-B2 Petrolatum-based compositions and methods of treatment for onychomycosis GLOBAL HEALTH SOLUTIONS LLC 2025-10-07 US claimed
US-5696164-A APPLYING MIXTURE OF UREA AND SULFHYDRYL-CONTAINING AMINO COMPOUND BY USING BANDAGE HAVING NAIL SHAPED CAVITY JOHNSON & JOHNSON CONSUMER PRODUCTS, INC. (US) 1997-12-09 US claimed
EP-0755675-B1 Dermatological and/or pharmaceutical composition, process of preparation and utilization OREAL (FR) 1997-09-17 EP claimed
EP-0792137-A1 ANTIFUNGAL TREATMENT OF NAILS JOHNSON & JOHNSON CONSUMER PRODUCTS, INC. (US) 1997-09-03 EP claimed
WO-1997009973-A2 PERIPHERALLY ACTIVE ANTI-HYPERALGESIC OPIATES THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1997-03-20 WO claimed
WO-1996036739-A1 COMBINATIONS OF ACTIVE SUBSTANCES BAYER AKTIENGESELLSCHAFT (DE) 1996-11-21 WO claimed
WO-1996019186-A1 ANTIFUNGAL TREATMENT OF NAILS JOHNSON & JOHNSON CONSUMER PRODUCTS, INC. (US) 1996-06-27 WO claimed
US-5407663-A Swishing solution in mouth, expectorating EISEN DRORE (US) 1995-04-18 US claimed
EP-0389778-B1 Nail Varnish HOFFMANN LA ROCHE (CH) 1994-05-04 EP claimed
EP-0024334-B1 MORPHOLINE DERIVATIVES, PROCESS FOR THEIR PRODUCTION, PHARMACEUTICAL PREPARATIONS CONTAINING THESE DERIVATIVES F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1983-07-20 EP claimed
EP-0024334-A1 Morpholine derivatives, process for their production, pharmaceutical preparations containing these derivatives F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1981-03-04 EP claimed