SCHEMBL15071204

SCHEMBL15071204

Cc1nc2cncc(C#N)c2[nH]1

nearest known ligand 0.32

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 1/20 0.32
CYP11B1 P15538 3/20 0.32
CYP11B2 P19099 3/20 0.32
KDM5A P29375 1/20 0.31
CLK1 P49759 2/20 0.30
CDK5 Q00535 2/20 0.30
DYRK1A Q13627 2/20 0.30
CDK5R1 Q15078 2/20 0.30
CLK2 P49760 1/20 0.30
CLK3 P49761 1/20 0.30
CLK4 Q9HAZ1 1/20 0.30
DYRK1B Q9Y463 1/20 0.30
GAA P10253 1/20 0.30
PRKCQ Q04759 1/20 0.30
PRKCD Q05655 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21263268 0.75 PARP1 (0.41) DYRK1AGAA
SCHEMBL15812731 0.74 CSNK1A1 (0.33) ADORA3KDM5A
SCHEMBL15071082 0.72 CSNK2A1 (0.39) ADORA3
SCHEMBL15334774 0.67 TSHR (0.44) CYP11B1CYP11B2PRKCQPRKCD
SCHEMBL11296434 0.67 KDM4A (0.33)
SCHEMBL27185599 0.67 HSP90AA1 (0.41) KDM5A
SCHEMBL30951806 0.66 PARP1 (0.43) CLK1CDK5DYRK1ACDK5R1CLK4
SCHEMBL9615544 0.66 ALDH1A1 (0.49) GAA
SCHEMBL24709786 0.64 CSNK1D (0.34) ADORA3CYP11B1CYP11B2
SCHEMBL21400917 0.64 KDM4E (0.40) KDM5AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013092940-A1 2, 4-DIAMINE-PYRIMIDINE DERIVATIVE AS SERINE/THREONINE KINASE INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2013-06-27 WO disclosed