SCHEMBL15071404

SCHEMBL15071404

O=C/C=C/C1NCCc2cc(Cl)ccc21

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 7/20 0.44
HTR2A P28223 6/20 0.44
HTR2B P41595 6/20 0.44
KDM1A O60341 2/20 0.40
SRD5A1 P18405 4/20 0.38
PNMT P11086 1/20 0.37
PRCP P42785 1/20 0.36
ADRB1 P08588 1/20 0.36
HTR1A P08908 1/20 0.36
ADRA2A P08913 1/20 0.36
ADRA2B P18089 1/20 0.36
ADRA2C P18825 1/20 0.36
CNR1 P21554 1/20 0.36
SLC6A2 P23975 1/20 0.36
SLC6A4 P31645 1/20 0.36
HRH1 P35367 1/20 0.36
KCNH2 Q12809 1/20 0.36
F7 P08709 1/20 0.35
PARP1 P09874 1/20 0.35
F3 P13726 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27343433 0.85 HTR2C (0.49) HTR2CHTR2AHTR2BKDM1ASRD5A1
SCHEMBL28823682 0.77 HTR2C (0.43) HTR2CHTR2AHTR2BKDM1ASRD5A1
SCHEMBL27919507 0.73 HTR2C (0.50) HTR2CHTR2AHTR2BKDM1APNMT
SCHEMBL31579647 0.70 HTR2A (0.61) HTR2CHTR2AHTR2BKDM1AADRB1
SCHEMBL6159366 0.70 HTR2A (0.61) HTR2CHTR2AHTR2BKDM1AADRB1
SCHEMBL27818616 0.70 CA1 (0.50) KDM1ASLC6A9
SCHEMBL27975547 0.69 PNMT (0.41) HTR2CHTR2AHTR2BSRD5A1PNMT
SCHEMBL15568933 0.69 TSHR (0.60) HTR2CHTR2AHTR2BKDM1ASRD5A1
SCHEMBL15071424 0.69 ALDH1A1 (0.52) HTR2CHTR2AHTR2BKDM1AOPRM1
SCHEMBL8222482 0.67 PRCP (0.67) HTR2CHTR2AKDM1APRCP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013096150-A1 SUBSTITUTED PIPERIDINES AS HDM2 INHIBITORS MERCK SHARP & DOHME CORP. (US) 2013-06-27 WO disclosed