SCHEMBL1507792

SCHEMBL1507792

N#Cc1ccc(Cn2ccnc2Sc2ccccc2)cc1

nearest known ligand 0.56

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.56
MEN1 O00255 2/20 0.56
ALDH1A1 P00352 3/20 0.49
CYP1A2 P05177 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2D6 P10635 1/20 0.49
CYP2C9 P11712 1/20 0.49
ALOX12 P18054 1/20 0.49
CYP2C19 P33261 1/20 0.49
MAOA P21397 1/20 0.47
MAOB P27338 1/20 0.47
CYP11B1 P15538 3/20 0.46
CYP11B2 P19099 3/20 0.46
CYP19A1 P11511 6/20 0.46
HTT P42858 2/20 0.43
MAPT P10636 1/20 0.43
LMNA P02545 1/20 0.43
HPGD P15428 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL1507763 0.80 CYP19A1 (0.49) KMT2AMEN1ALDH1A1CYP1A2CYP3A4
SCHEMBL10424264 0.77 ALDH1A1 (0.58) KMT2AMEN1ALDH1A1HTTLMNA
SCHEMBL1507751 0.77 CYP11B1 (0.56) CYP11B1CYP11B2CYP19A1
SCHEMBL30610947 0.76 CYP11B1 (0.48) KMT2AMEN1ALDH1A1CYP1A2CYP3A4
SCHEMBL1507873 0.76 CYP11B1 (0.48) KMT2AMEN1ALDH1A1CYP1A2CYP3A4
SCHEMBL8541839 0.75 KMT2A (0.50) KMT2AMEN1ALDH1A1CYP1A2CYP3A4
Hydrochloric Acid SCHEMBL1507947 0.75 CYP11B1 (0.47) KMT2AMEN1ALDH1A1CYP1A2CYP3A4
SCHEMBL22782676 0.74 LIMK2 (0.55) MAOBCYP11B1CYP11B2CYP19A1
SCHEMBL7855826 0.73 LMNA (0.59) KMT2ACYP11B1CYP11B2CYP19A1LMNA
SCHEMBL10425588 0.73 CYP19A1 (0.51) KMT2ACYP11B1CYP11B2CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0236940-B3 Alpha-heterocycle substituted tolunitriles NOVARTIS AG (CH) 2011-03-23 EP disclosed
US-5473078-A Aromatase inhibiting compounds CIBA-GEIGY CORPORATION (US) 1995-12-05 US disclosed
US-5352795-A Condensing triazolylmethylbenzonitrile with fluorobenzonitrile under basic conditions using alkali metal alkoxide CIBA-GEIGY CORPORATION (US) 1994-10-04 US disclosed
EP-0236940-B1 ALPHA-HETEROCYCLE SUBSTITUTED TOLUNITRILES CIBA-GEIGY AG (CH) 1993-09-22 EP disclosed
US-5112845-A Inhibitors of estrogen synthesis, veterinary medicine CIBA-GEIGY CORPORATION (US) 1992-05-12 US disclosed
US-5071861-A Aromatase enzyme inhibitor; antiestrogens CIBA-GEIGY CORPORATION (US) 1991-12-10 US disclosed
US-4978672-A Alpha-heterocyclc substituted tolunitriles CIBA-GEIGY CORPORATION (US) 1990-12-18 US disclosed
US-4937250-A AROMATASE ENZYME INHIBITORS CIBA-GEIGY CORPORATION (US) 1990-06-26 US disclosed
US-4749713-A Alpha-heterocycle substituted tolunitriles CIBA-GEIGY CORPORATION (US) 1988-06-07 US disclosed
EP-0236940-A2 Alpha-heterocycle substituted tolunitriles CIBA-GEIGY AG (CH) 1987-09-16 EP disclosed