SCHEMBL1508874

SCHEMBL1508874

CC1(c2ccc(Cl)nc2)NS(=O)(=O)NC1c1ccc(C(F)(F)F)c(F)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNQ3 O43525 2/20 0.39
KCNQ2 O43526 2/20 0.39
KCNE1 P15382 2/20 0.39
KCNQ1 P51787 2/20 0.39
CHRM2 P08172 1/20 0.37
DRD2 P14416 1/20 0.37
CHRNB2 P17787 1/20 0.37
DRD4 P21917 1/20 0.37
CHRNB4 P30926 1/20 0.37
CHRNA3 P32297 1/20 0.37
DRD3 P35462 1/20 0.37
CHRNA7 P36544 1/20 0.37
CHRNA4 P43681 1/20 0.37
TMEM97 Q5BJF2 1/20 0.37
KDM1A O60341 1/20 0.35
HDAC3 O15379 1/20 0.32
HDAC1 Q13547 1/20 0.32
HDAC2 Q92769 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32
CYP11B1 P15538 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1508873 0.89 KCNQ3 (0.39) KCNQ3KCNQ2KCNE1KCNQ1CHRM2
SCHEMBL7921145 0.87 MDM2 (0.36) KCNQ3KCNQ2KCNE1KCNQ1
SCHEMBL1508741 0.87 MDM2 (0.36) KCNQ3KCNQ2KCNE1KCNQ1
SCHEMBL14793575 0.80 KMT2A (0.33) KCNQ3KCNQ2KCNE1KCNQ1CHRNB2
SCHEMBL14817142 0.80 KMT2A (0.33) KCNQ3KCNQ2KCNE1KCNQ1CHRNB2
SCHEMBL1508733 0.78 KMO (0.32)
SCHEMBL1508742 0.76 KCNQ3 (0.34) KCNQ3KCNQ2KCNE1KCNQ1
SCHEMBL1508739 0.76 KCNQ3 (0.34) KCNQ3KCNQ2KCNE1KCNQ1
SCHEMBL1509045 0.75 KCNQ3 (0.31) KCNQ3KCNQ2KCNE1KCNQ1
SCHEMBL1509102 0.71 TAAR1 (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2298778-A1 IMIDAZOTHIAZOLE DERIVATIVE HAVING 4,7-DIAZASPIROÝ2.5¨OCTANE RING STRUCTURE Daiichi Sankyo Company, Limited (JP) 2011-03-23 EP disclosed
WO-2009151069-A1 IMIDAZOTHIAZOLE DERIVATIVE HAVING 4,7-DIAZASPIRO[2.5]OCTANE RING STRUCTURE 第一三共株式会社 (JP) 2009-12-17 WO disclosed