SCHEMBL1509079

SCHEMBL1509079

COc1cc([C@H]2NC(=S)N[C@@]2(C)c2ccc(Cl)nc2)ccc1Cl

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 2/20 0.34
ADAM17 P78536 1/20 0.33
ADAMTS5 Q9UNA0 1/20 0.33
ALDH1A1 P00352 7/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
NPC1 O15118 1/20 0.32
POLB P06746 1/20 0.32
RAB9A P51151 1/20 0.32
GAA P10253 2/20 0.32
KCNQ3 O43525 1/20 0.32
KCNQ2 O43526 1/20 0.32
GRM4 Q14833 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32
MAPK1 P28482 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
MAPT P10636 2/20 0.31
LMNA P02545 1/20 0.31
CHRNB2 P17787 1/20 0.31
CHRNB4 P30926 1/20 0.31
CHRNA3 P32297 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1508909 0.86 KCNQ3 (0.37) KCNQ3KCNQ2CHRNB2CHRNB4CHRNA3
SCHEMBL3831124 0.83 NPSR1 (0.34) ALDH1A1SMN1; SMN2KCNQ3KCNQ2LMNA
SCHEMBL3831127 0.83 NPSR1 (0.34) ALDH1A1SMN1; SMN2KCNQ3KCNQ2LMNA
SCHEMBL2487546 0.83 NPSR1 (0.34) ALDH1A1SMN1; SMN2KCNQ3KCNQ2LMNA
SCHEMBL1508736 0.80 NPC1 (0.34) PDE10AADAM17ADAMTS5NPC1POLB
SCHEMBL1508733 0.78 KMO (0.32) PDE10AADAM17ADAMTS5ALDH1A1NPC1
SCHEMBL3827291 0.78 NPSR1 (0.36) ALDH1A1SMN1; SMN2KCNQ3KCNQ2CHRNB2
SCHEMBL3833887 0.78 NPSR1 (0.36) ALDH1A1SMN1; SMN2KCNQ3KCNQ2CHRNB2
SCHEMBL7943091 0.74 ALDH1A1 (0.31) ALDH1A1MAPT
SCHEMBL1508787 0.70 NPSR1 (0.36) ALDH1A1GAAMAPTLMNACHRNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2298778-A1 IMIDAZOTHIAZOLE DERIVATIVE HAVING 4,7-DIAZASPIROÝ2.5¨OCTANE RING STRUCTURE Daiichi Sankyo Company, Limited (JP) 2011-03-23 EP disclosed