SCHEMBL1509205

SCHEMBL1509205

NC(=O)c1nc(NC=O)c[nH]1

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3317344 0.72 ALDH1A1 (0.32)
SCHEMBL28875234 0.71
SCHEMBL3821371 0.70 LMNA (0.41)
SCHEMBL965458 0.69 LMNA (0.34)
SCHEMBL8561 0.69
SCHEMBL161337 0.69
SCHEMBL161336 0.69
SCHEMBL1857158 0.67
SCHEMBL24294078 0.67
SCHEMBL10861571 0.67 PARP1 (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2295976-A1 Markers for colorectal cancer Auvation Ltd (GB) 2011-03-16 EP disclosed
US-20100216156-A1 CANCER MARKERS MURRAY GRAEME IAN 2010-08-26 US disclosed
EP-0405370-B2 Riboflavinoverproducing strains of bacteria DSM IP ASSETS BV (NL) 2007-12-19 EP disclosed
US-7091000-B2 Bacterial strains which overproduce riboflavin and methods of use thereof DSM NUTRITIONAL PRODUCTS, INC. (US) 2006-08-15 US disclosed
US-20030232406-A1 Bacterial strains which overproduce riboflavin ROCHE VITAMINS, INC. 2003-12-18 US disclosed
US-6551813-B1 Yeast extract, glucose, a magnesium salt, a manganese salt, a calcium salt, an iron salt, a phosphate buffer, and additional salt selected from the group consisting of a glutamic acid salt, a citric acid salt, and a succinic acid salt ROCHE VITAMINS INC. 2003-04-22 US disclosed
US-6322995-B1 RECOMBINANT GRAM POSITIVE BACTERIUM USED FOR PRODUCING RIBOFLAVIN F. HOFFMANN-LA ROCHE AG (CH) 2001-11-27 US disclosed
EP-0405370-B1 Riboflavinoverproducing strains of bacteria HOFFMANN LA ROCHE (CH) 2000-08-30 EP disclosed
EP-1001026-A2 Riboflavinoverproducing strains of bacteria F. Hoffmann-La Roche AG (CH) 2000-05-17 EP disclosed
US-5925538-A CULTURING RECOMBINANT BACTERIUM HAVING EXOGENOUS NUCLEIC ACID SEQUENCE CODING FOR PROMOTER AND OPEN READING FRAME 3 STRUCTURAL GENE SIMILAR TO A BACILLUS SUBTILIS RIBOFLAVIN OPERON GENE, RECOVERING AT LEAST 10 GRAMS PER LITER ROCHE VITAMINS INC. (US) 1999-07-20 US disclosed
US-5837528-A NUCLEOTIDE SEQUENCE OF RIB OPERON AND ITS OPEN READING FRAMES; GENETIC ENGINEERING HOFFMANN LA ROCHE, INC. (US) 1998-11-17 US disclosed
US-5800979-A Gas chromatography/mass spectrometric determination of folic acid coenzymes KOLHOUSE J FRED (US) 1998-09-01 US disclosed
EP-0405370-A1 Riboflavinoverproducing strains of bacteria F. HOFFMANN-LA ROCHE AG (CH) 1991-01-02 EP disclosed