SCHEMBL1515134

SCHEMBL1515134

COc1cccc(C2CC2)c1

nearest known ligand 0.77

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 4/20 0.77
DRD2 P14416 2/20 0.64
ADRA1A P35348 5/20 0.56
HTR1A P08908 3/20 0.56
ADRA1D P25100 3/20 0.56
ADRA1B P35368 3/20 0.56
HTR2A P28223 2/20 0.53
HTR2B P41595 2/20 0.53
DDB1 Q16531 1/20 0.51
CRBN Q96SW2 1/20 0.51
GID4 Q8IVV7 1/20 0.51
KDM1A O60341 1/20 0.49
RCOR1 Q9UKL0 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30997824 1.00 HTR2C (0.77) HTR2CDRD2ADRA1AHTR1AADRA1D
Methyl Alcohol SCHEMBL8097139 0.96 HTR2C (0.72) HTR2CDRD2ADRA1AHTR1AADRA1D
SCHEMBL28695004 0.93 HTR2C (0.68) HTR2CDRD2ADRA1AHTR1AADRA1D
SCHEMBL7844832 0.92 HTR2C (0.72) HTR2CDRD2ADRA1AHTR1AADRA1D
SCHEMBL1515075 0.92 HTR2C (0.72) HTR2CDRD2ADRA1AHTR1AADRA1D
SCHEMBL28695001 0.91 HTR2C (0.66) HTR2CDRD2ADRA1AHTR1AADRA1D
Ethylamine SCHEMBL8089244 0.91 HTR2C (0.66) HTR2CDRD2ADRA1AHTR1AADRA1D
SCHEMBL7215877 0.91 HTR2C (0.66) HTR2CDRD2ADRA1AHTR1AADRA1D
Ammonia Solution, Strong SCHEMBL19664329 0.90 HTR2C (0.70) HTR2CDRD2ADRA1AHTR1AADRA1D
SCHEMBL2095198 0.90 HTR2C (0.70) HTR2CDRD2ADRA1AHTR1AADRA1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 51 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3363788-A1 CANNABINOID RECEPTOR MODULATORS Arena Pharmaceuticals, Inc. (US) 2018-08-22 EP claimed
US-20130165412-A1 CANNABINOID RECEPTOR MODULATORS ARENA PHARMACEUTICALS, INC. 2013-06-27 US claimed
US-20120214766-A1 CANNABINOID RECEPTOR MODULATORS ARENA PHARMACEUTICALS, INC. 2012-08-23 US claimed
EP-2470508-A1 CANNABINOID RECEPTOR MODULATORS Arena Pharmaceuticals, Inc. (US) 2012-07-04 EP claimed
WO-2011025541-A1 CANNABINOID RECEPTOR MODULATORS ARENA PHARMACEUTICALS, INC. (US) 2011-03-03 WO claimed
US-11771695-B2 Cannabinoid receptor modulators ARENA PHARMACEUTICALS, INC. (US) 2023-10-03 US disclosed
US-11746091-B2 Cannabinoid receptor modulators ARENA PHARMACEUTICALS, INC. (US) 2023-09-05 US disclosed
EP-3798217-B1 PIPERIDINE CXCR7 RECEPTOR MODULATORS IDORSIA PHARMACEUTICALS LTD (CH) 2023-02-22 EP disclosed
CN-110563717-B Piperidine CXCR7 receptor modulators 爱杜西亚药品有限公司 2022-08-09 CN disclosed
CN-109563085-B Piperidine CXCR7 receptor modulators 爱杜西亚药品有限公司 2022-08-09 CN disclosed
US-20220241274-A1 CANNABINOID RECEPTOR MODULATORS ARENA PHARMACEUTICALS, INC. 2022-08-04 US disclosed
CN-109970708-B Cannabinoid receptor modulators 艾尼纳制药公司 2022-06-21 CN disclosed
WO-2012116278-A1 CANNABINOID RECEPTOR MODULATORS ARENA PHARMACEUTICALS, INC. (US) 2012-08-30 WO disclosed
WO-2012116279-A1 CANNABINOID RECEPTOR MODULATORS ARENA PHARMACEUTICALS, INC. (US) 2012-08-30 WO disclosed
US-20120214766-A1 CANNABINOID RECEPTOR MODULATORS ARENA PHARMACEUTICALS, INC. 2012-08-23 US disclosed
EP-2470508-A1 CANNABINOID RECEPTOR MODULATORS Arena Pharmaceuticals, Inc. (US) 2012-07-04 EP disclosed
US-7977322-B2 Such as 1-Benzo[1,3]dioxol-5-yl-cyclopropanecarboxylic acid [5-(2-methoxy-pyridin-3-ylmethyl)-thiazol-2-yl]-amide 5-(2-Methoxy-pyridin-3-ylmethyl)-thiazol-2-ylamine; cystic fibrosis transmembrane conductance regulator disorders VERTEX PHARMACEUTICALS INCORPORATED (US) 2011-07-12 US disclosed
WO-2011025541-A1 CANNABINOID RECEPTOR MODULATORS ARENA PHARMACEUTICALS, INC. (US) 2011-03-03 WO disclosed
US-5051447-A Applying aromatic oximes to plants, seeds or soils BASF AKTIENGESELLSCHAFT (DE) 1991-09-24 US disclosed
US-4952720-A Ortho-substituted benzyl carboxylates and fungicides which contain these compounds BASF AKTIENGSELLSCHAFT (DE) 1990-08-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120214766-A1 CANNABINOID RECEPTOR MODULATORS CNR1, CNR2, TRPV1 HTR2C 711/4885DRD2 1476/4885ADRA1A 195/4885
US-11746091-B2 Cannabinoid receptor modulators CNR1, CNR2, TRPV1 HTR2C 711/4885DRD2 1476/4885ADRA1A 195/4885
US-20220241274-A1 CANNABINOID RECEPTOR MODULATORS CNR2, CNR1, OPRL1 HTR2C 78/4885DRD2 669/4885ADRA1A 93/4885
US-11771695-B2 Cannabinoid receptor modulators CNR2, CNR1, OPRL1 HTR2C 78/4885DRD2 669/4885ADRA1A 93/4885
US-20130165412-A1 CANNABINOID RECEPTOR MODULATORS CNR1, CNR2, TRPV1 HTR2C 711/4885DRD2 1476/4885ADRA1A 195/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.