SCHEMBL15210210

SCHEMBL15210210

c1ccc(OCc2cc[nH]n2)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.57
CYSLTR2 Q9NS75 1/20 0.49
CYSLTR1 Q9Y271 1/20 0.49
KCNA3 P22001 1/20 0.46
MAPT P10636 2/20 0.46
MAOA P21397 1/20 0.43
MAOB P27338 1/20 0.43
NISCH Q9Y2I1 1/20 0.43
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
CYP19A1 P11511 2/20 0.42
TP53 P04637 1/20 0.42
TSHR P16473 1/20 0.42
APP P05067 1/20 0.41
ALOX15 P16050 1/20 0.41
NOS1 P29475 1/20 0.40
ALDH1A1 P00352 1/20 0.40
LMNA P02545 1/20 0.40
HPGD P15428 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9721057 0.93 LTA4H (0.52) KCNH2CYSLTR2CYSLTR1KCNA3MAPT
SCHEMBL7207747 0.81 KCNH2 (0.36) KCNH2CYSLTR2CYSLTR1MAPTSMN1; SMN2
SCHEMBL26497069 0.81 SMN1; SMN2 (0.49) KCNH2MAOBNPC1RAB9ASMN1; SMN2
SCHEMBL30298095 0.76 NPC1 (0.45) NPC1ALDH1A1GRM5
SCHEMBL27733181 0.74 TSHR (0.58) NPC1RAB9ASMN1; SMN2TSHR
SCHEMBL5755405 0.73 KCNH2 (0.30) KCNH2
SCHEMBL12042914 0.73 KCNH2 (0.58) KCNH2CYSLTR2CYSLTR1MAPTNPC1
SCHEMBL6445371 0.71 KCNH2 (0.67) KCNH2CYSLTR2CYSLTR1KCNA3MAOB
SCHEMBL2288762 0.71 CALM1 (0.46) RAB9ASMN1; SMN2TSHRALDH1A1HPGD
SCHEMBL4427549 0.71 KCNH2 (0.55) KCNH2CYSLTR2CYSLTR1KCNA3MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230322744-A1 COMPOUNDS AS GLP-1R AGONISTS TERNS PHARMACEUTICALS, INC. 2023-10-12 US disclosed
US-20230322744-A1 COMPOUNDS AS GLP-1R AGONISTS TERNS PHARMACEUTICALS, INC. 2023-10-12 US disclosed
US-20230322744-A1 COMPOUNDS AS GLP-1R AGONISTS TERNS PHARMACEUTICALS, INC. 2023-10-12 US disclosed
CN-116507326-A Compounds as GLP-1R agonists 拓臻制药公司 2023-07-28 CN disclosed
EP-4199919-A1 COMPOUNDS AS GLP-1R AGONISTS Terns Pharmaceuticals, Inc. (US) 2023-06-28 EP disclosed
US-20220089578-A1 COMPOUNDS AS GLP-1R AGONISTS TERNS PHARMACEUTICALS, INC. 2022-03-24 US disclosed
WO-2022040600-A1 COMPOUNDS AS GLP-1R AGONISTS TERNS PHARMACEUTICALS, INC. (US) 2022-02-24 WO disclosed
WO-2022040600-A1 COMPOUNDS AS GLP-1R AGONISTS TERNS PHARMACEUTICALS, INC. (US) 2022-02-24 WO disclosed
CN-104271595-B Proteins toxic to hemipteran insect species 孟山都技术公司 2018-09-18 CN disclosed
US-20130226549-A1 STRUCTURE-BASED FRAGMENT HOPPING FOR LEAD OPTIMIZATION AND IMPROVEMENT IN SYNTHETIC ACCESSIBILITY TSENG, YUFENG J. (TW) 2013-08-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230322744-A1 COMPOUNDS AS GLP-1R AGONISTS GLP1R, GIPR, GCGR KCNH2 3089/4885CYSLTR2 1419/4885CYSLTR1 924/4885
US-20220089578-A1 COMPOUNDS AS GLP-1R AGONISTS GLP1R, GIPR, GCGR KCNH2 3089/4885CYSLTR2 1419/4885CYSLTR1 924/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.