SCHEMBL6445371

SCHEMBL6445371

c1ccc(OCc2ccccn2)cc1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.67
ALDH1A1 P00352 2/20 0.66
SMN1; SMN2 Q16637 2/20 0.66
KDM4E B2RXH2 1/20 0.66
PARP10 Q53GL7 1/20 0.62
CYP1A2 P05177 1/20 0.57
CYP3A4 P08684 1/20 0.57
CYP2D6 P10635 1/20 0.57
CYP2C9 P11712 1/20 0.57
ABCB1 P08183 1/20 0.53
HTR1A P08908 1/20 0.53
DRD2 P14416 1/20 0.53
CYSLTR2 Q9NS75 1/20 0.52
CYSLTR1 Q9Y271 1/20 0.52
FFAR1 O14842 1/20 0.51
HPGD P15428 1/20 0.50
TLR4 O00206 1/20 0.50
TLR2 O60603 1/20 0.50
MEN1 O00255 1/20 0.50
KMT2A Q03164 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10388636 0.92 KDM4E (0.63) KCNH2ALDH1A1SMN1; SMN2KDM4EPARP10
SCHEMBL1312722 0.88 SMN1; SMN2 (0.62) KCNH2ALDH1A1SMN1; SMN2KDM4EPARP10
SCHEMBL22874534 0.86 PARP10 (0.66) KCNH2ALDH1A1SMN1; SMN2KDM4EPARP10
SCHEMBL5667052 0.84 KDM4E (0.63) KCNH2ALDH1A1SMN1; SMN2KDM4EPARP10
SCHEMBL22967393 0.84 ALDH1A1 (0.63) ALDH1A1SMN1; SMN2KDM4EPARP10CYP1A2
SCHEMBL17712563 0.84 SMN1; SMN2 (0.63) KCNH2ALDH1A1SMN1; SMN2KDM4EPARP10
SCHEMBL21568937 0.84 KDM4E (0.63) KCNH2ALDH1A1SMN1; SMN2KDM4EPARP10
SCHEMBL864159 0.84 KDM4E (0.58) KCNH2ALDH1A1SMN1; SMN2KDM4EPARP10
SCHEMBL1073540 0.84 SYK (0.68) ALDH1A1SMN1; SMN2KDM4EPARP10CYP1A2
SCHEMBL169753 0.84 SMN1; SMN2 (0.63) ALDH1A1SMN1; SMN2KDM4EPARP10CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 53 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100383138-C N-monoacetyl o-phenylenediamines, their fused heterocyclic derivatives and their use as medicaments HOFFMANN LA ROCHE (CH) 2008-04-23 CN claimed
CN-1747948-A Novel n-monoacylated o-phenylenediamines, their condensed heterocyclic derivatives and their use as pharmaceutical agents HOFFMANN LA ROCHE (CH) 2006-03-15 CN claimed
US-6156774-A Beta-thiopropionyl-amino acid derivatives and their use as beta-lactamase inhibitors SMITHKLINE BEECHAM P.L.C. (GB) 2000-12-05 US claimed
EP-1000024-A1 MERCAPTOACYLAMINO ACIDS AS METALLO-BETA-LACTAMASE INHIBITORS SMITHKLINE BEECHAM PLC (GB) 2000-05-17 EP claimed
EP-0970062-A2 PYRROLIDINE AND THIAZOLE DERIVATIVES WITH METALLO-BETA-LACTAMASE INHIBITORY PROPERTIES SMITHKLINE BEECHAM PLC (GB) 2000-01-12 EP claimed
WO-1999006365-A1 MERCAPTOACYLAMINO ACIDS AS METALLO-BETA-LACTAMASE INHIBITORS SMITHKLINE BEECHAM PLC (GB) 1999-02-11 WO claimed
WO-1998040056-A2 PYRROLIDINE AND THIAZOLE DERIVATIVES WITH METALLO-BETA-LACTAMASE INHIBITORY PROPERTIES SMITHKLINE BEECHAM PLC (GB) 1998-09-17 WO claimed
US-5468721-A FOR CONTROLLING OR KILLING WEEDS MITSUBISHI PETROCHEMICAL CO., LTD. (JP) 1995-11-21 US claimed
CN-116063226-B Ether compound containing monoterpene phenol structure 云南省农业科学院茶叶研究所 2023-06-02 CN disclosed
CN-116063226-B Ether compound containing monoterpene phenol structure 云南省农业科学院茶叶研究所 2023-06-02 CN disclosed
CN-116063226-A Ether compound containing monoterpene phenol structure 云南省农业科学院茶叶研究所 2023-05-05 CN disclosed
CN-116063226-A Ether compound containing monoterpene phenol structure 云南省农业科学院茶叶研究所 2023-05-05 CN disclosed
WO-2023062627-A1 HERBICIDES AND USE THEREOF PROJINI AGCHEM LTD (IL) 2023-04-20 WO disclosed
US-20220196685-A1 PROBES FOR DETECTION OF COPPER THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2022-06-23 US disclosed
WO-1998017639-A1 BETA-THIOPROPIONYL-AMINO ACID DERIVATIVES AND THEIR USE AS BETA-LACTAMASE INHIBITORS SMITHKLINE BEECHAM PLC (GB) 1998-04-30 WO disclosed
US-4839369-A ANTIINFLAMMATORY AGENTS; ANTIALLERGENS RORER PHARMACEUTICAL CORPORATION (US) 1989-06-13 US disclosed
US-4728668-A Aryl and heteroaryl ethers as agents for the treatment of hypersensitive ailments USV PHARMACEUTICAL CORPORATION (US) 1988-03-01 US disclosed
US-4725619-A Aryl and heteroaryl ethers as agents for the treatment of hypersensitive ailments USV PHARMACEUTICAL CORPORATION (US) 1988-02-16 US disclosed
US-4631287-A Aryl and heteroaryl ethers as agents for the treatment of hypersensitive ailments USV PHARMACEUTICAL CORP. (US) 1986-12-23 US disclosed
US-4243807-A CHEMICAL INTERMEDIATES FOR HYPOTENSIVE AGENTS BOEHRINGER MANNHEIM GMBH (DE) 1981-01-06 US disclosed