SCHEMBL15212927

SCHEMBL15212927

O=C(O)Cc1occ2c(Cl)c(O)ccc12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 2/20 0.40
MAPT P10636 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
ALOX15 P16050 1/20 0.38
HPGD P15428 3/20 0.36
HSD17B10 Q99714 3/20 0.36
LMNA P02545 2/20 0.36
TSHR P16473 2/20 0.36
KDM4E B2RXH2 2/20 0.36
GAA P10253 2/20 0.36
RGS12 O14924 1/20 0.36
POLB P06746 1/20 0.36
NFKB1 P19838 1/20 0.36
APEX1 P27695 1/20 0.36
THPO P40225 1/20 0.36
BLM P54132 1/20 0.36
GNAI1 P63096 1/20 0.36
PMP22 Q01453 1/20 0.36
HIF1A Q16665 1/20 0.36
TDP1 Q9NUW8 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15212923 0.81 MAPT (0.44) CA2MAPTSMN1; SMN2ALOX15HPGD
SCHEMBL15211231 0.73 SMN1; SMN2 (0.57) CA2MAPTSMN1; SMN2ALOX15KDM4E
SCHEMBL12474263 0.69 LCK (0.44) CA2MAPTSMN1; SMN2ALOX15HPGD
SCHEMBL6136983 0.66 AKR1B1 (0.52) CA2MAPTHPGDHSD17B10LMNA
SCHEMBL29051963 0.66 AKR1B1 (0.61) CA2MAPTHPGDHSD17B10LMNA
SCHEMBL1650809 0.66 KDM4E (0.50) HPGDHSD17B10LMNAKDM4EGAA
SCHEMBL2368215 0.65 CYP3A4 (0.55) HSD17B10TSHRALDH1A1MAPK1ESR1
SCHEMBL31266634 0.64 AKR1B1 (0.43) CA2MAPTSMN1; SMN2HPGDHSD17B10
SCHEMBL23191190 0.63 CYP3A4 (0.52) HSD17B10TSHRMAPK1ESR1ESR2
SCHEMBL9623621 0.62 CA1 (0.48) CA2MAPTSMN1; SMN2ALOX15HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2838891-A1 AROMATIC RING COMPOUND Takeda Pharmaceutical Company Limited (JP) 2015-02-25 EP disclosed
WO-2013125732-A1 AROMATIC RING COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2013-08-29 WO disclosed