Fumaric Acid

Fumaric Acid

SCHEMBL152140

CCCC[BiH]CCCC.O=C(O)C=CC(=O)O

nearest known ligand 0.50

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Known targets — ChEMBL curated mechanism

ACEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ATP4AATP4BAXLBTKCACNA1CCACNA1DCACNA1FCACNA1SCCR5CHRM2CHRM3CPT1BCPT2DPP4DRD1DRD2EGFRERBB2ERBB4FLT3HRH1HRH3HTR1AHTR2AHTR2BHTR2CHTR4JAK1JAK2JAK3KCNH2KMT2AMAP2K1MAP2K2MEN1MLNRMPLMTORPPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PLK4PPARGRENS1PR1SLC6A2SLC6A3SLC6A4SMOTYK2atpAatpBatpCatpDatpEatpFatpFHatpGpol

The experimentally established mechanism targets of Fumaric Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 5/20 0.50
TSHR P16473 2/20 0.43
TP53 P04637 1/20 0.43
EGLN1 Q9GZT9 1/20 0.43
EGLN3 Q9H6Z9 1/20 0.43
ACHE P22303 1/20 0.41
BACE1 P56817 1/20 0.41
PLA2G1B P04054 6/20 0.41
ATG4B Q9Y4P1 6/20 0.41
THRA P10827 1/20 0.40
THRB P10828 1/20 0.40
CYP1A2 P05177 1/20 0.40
TDP1 Q9NUW8 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Maleic Acid SCHEMBL11695225 0.82 HCAR2 (0.64) HCAR2TSHRTP53EGLN1EGLN3
Fumaric Acid SCHEMBL28133862 0.82 HCAR2 (0.64) HCAR2TSHRTP53EGLN1EGLN3
Octane SCHEMBL6872110 0.79 HCAR2 (0.65) HCAR2TSHRTDP1
Octane SCHEMBL6872114 0.79 HCAR2 (0.65) HCAR2TSHRTDP1
Fumaric Acid SCHEMBL3414625 0.79 HCAR2 (0.65) HCAR2TSHRTDP1
Octane SCHEMBL2904002 0.79 HCAR2 (0.65) HCAR2TSHRTDP1
Nonane SCHEMBL8691965 0.79 HCAR2 (0.65) HCAR2TSHRTDP1
Fumaric Acid SCHEMBL3414623 0.79 HCAR2 (0.65) HCAR2TSHRTDP1
Decane SCHEMBL9668679 0.79 HCAR2 (0.65) HCAR2TSHRTDP1
Octane SCHEMBL8193217 0.79 HCAR2 (0.65) HCAR2TSHRTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8563675-B2 Curable compositions composed of silanes with two hydrolyzable groups HENKEL AG & CO. KGAA (DE) 2013-10-22 US disclosed
US-20120059130-A1 CURABLE COMPOSITIONS CONSISTING OF SILANES WITH THREE HYDROLYSABLE GROUPS HENKEL AG & CO. KGAA (DE) 2012-03-08 US disclosed
US-20100216950-A1 CURABLE COMPOSITIONS CONSISTING OF SILANES WITH THREE HYDROLYSABLE GROUPS HENKEL AG & CO. KGAA (DE) 2010-08-26 US disclosed
US-20100204387-A1 CURABLE COMPOSITIONS COMPOSED OF SILANES WITH TWO HYDROLYZABLE GROUPS HENKEL AG & CO. KGAA (DE) 2010-08-12 US disclosed