SCHEMBL15214877

SCHEMBL15214877

Cc1cc(-c2cscc2C#N)ccc1O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AR P10275 4/20 0.46
TLR8 Q9NR97 3/20 0.39
HSD17B1 P14061 4/20 0.39
HSD17B2 P37059 4/20 0.39
PGR P06401 2/20 0.38
ESR2 Q92731 6/20 0.38
CYP3A4 P08684 3/20 0.38
CYP2D6 P10635 3/20 0.38
CYP2C19 P33261 3/20 0.38
ESR1 P03372 5/20 0.38
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
CYP1A2 P05177 1/20 0.37
MAPT P10636 1/20 0.37
G6PD P11413 1/20 0.37
CYP2C9 P11712 1/20 0.37
PKM P14618 1/20 0.37
HPGD P15428 1/20 0.37
ALOX15 P16050 1/20 0.37
ALOX12 P18054 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3139052 0.78 ALOX15 (0.48) ARPGRESR2CYP3A4ESR1
SCHEMBL3320197 0.78 CYP2A6 (0.43) ARPGRESR2CYP3A4CYP2D6
SCHEMBL7388799 0.76 PTGS2 (0.47) ARESR2CYP3A4CYP2C19ESR1
SCHEMBL2474861 0.76 ESR2 (0.63) ARESR2ESR1
SCHEMBL29084993 0.73 AR (0.47) ARHSD17B1HSD17B2ESR2CYP3A4
SCHEMBL29084999 0.72 AR (0.46) ARHSD17B1HSD17B2ESR2CYP3A4
SCHEMBL20056706 0.71 AR (0.51) ARTLR8HSD17B1HSD17B2ESR2
SCHEMBL30536525 0.71 ESR2 (0.48) ARHSD17B1HSD17B2ESR2CYP3A4
SCHEMBL2786046 0.69 AR (0.57) ARHSD17B1HSD17B2ESR2ALDH1A1
SCHEMBL272034 0.69 HSD17B1 (0.68) ARHSD17B1HSD17B2ESR2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9067928-B2 Compounds and methods of use ABBVIE INC. (US) 2015-06-30 US disclosed
EP-2376085-B1 COMPOUNDS AND METHODS OF USE GENENTECH INC (US) 2014-02-26 EP disclosed
US-8518970-B2 Compounds and methods of use ABBVIE INC. (US) 2013-08-27 US disclosed