SCHEMBL15219409

SCHEMBL15219409

N#COc1cccc(CN=N)c1

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
F2 P00734 6/20 0.34
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
TAAR1 Q96RJ0 3/20 0.32
IDO1 P14902 2/20 0.32
AGXT P21549 2/20 0.32
P2RX7 Q99572 1/20 0.32
CYP1A1 P04798 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP1B1 Q16678 1/20 0.32
RAB9A P51151 1/20 0.32
MIF P14174 1/20 0.31
GRIN1 Q05586 2/20 0.31
GRIN2B Q13224 2/20 0.31
GRIN2D O15399 1/20 0.31
GRIN3B O60391 1/20 0.31
GRIN2A Q12879 1/20 0.31
GRIN2C Q14957 1/20 0.31
GRIN3A Q8TCU5 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14340523 0.80 FFAR1 (0.41) F2MEN1KMT2A
SCHEMBL158382 0.80 CHRM2 (0.38) MEN1KMT2ATAAR1IDO1AGXT
SCHEMBL15219801 0.77 TAAR1 (0.55) TAAR1IDO1AGXTGRIN1GRIN2B
SCHEMBL14730561 0.77 TSHR (0.44) MEN1KMT2A
SCHEMBL28286056 0.77 PNMT (0.44) TAAR1IDO1AGXT
SCHEMBL10835184 0.76 ALDH1A1 (0.39) MEN1KMT2AIDO1AGXTCYP1A2
SCHEMBL28114320 0.75 IDO1 (0.41) F2MEN1KMT2AIDO1AGXT
SCHEMBL26009 0.74 KMT2A (0.41) MEN1KMT2ACYP1A1CYP1A2CYP1B1
SCHEMBL20350466 0.72 TAAR1 (0.49) TAAR1IDO1AGXT
SCHEMBL23776528 0.71 HRH3 (0.47)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2631238-A1 Spirocyclic inhibitors of serine proteases for the treatment of hcv infections VERTEX PHARMACEUTICALS INCORPORATED (US) 2013-08-28 EP disclosed