SCHEMBL15224432

SCHEMBL15224432

O=C(O)N1CCN(Cc2cncc(Br)c2)CC1

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.51
ALDH1A1 P00352 5/20 0.51
HTT P42858 2/20 0.51
FAAH O00519 3/20 0.45
LMNA P02545 2/20 0.44
HPGD P15428 1/20 0.44
NPSR1 Q6W5P4 1/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
MAPT P10636 1/20 0.42
PRKAB2 O43741 1/20 0.41
PRKAG1 P54619 1/20 0.41
PRKAA2 P54646 1/20 0.41
PRKAA1 Q13131 1/20 0.41
PRKAG3 Q9UGI9 1/20 0.41
PRKAG2 Q9UGJ0 1/20 0.41
PRKAB1 Q9Y478 1/20 0.41
GPR183 P32249 1/20 0.41
POLB P06746 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27881616 0.87 KDM4E (0.47) KDM4EALDH1A1HTTFAAHLMNA
SCHEMBL15205816 0.82 KDM4E (0.44) KDM4EALDH1A1HTTFAAHNPSR1
SCHEMBL4757751 0.82 KDM4E (0.51) KDM4EALDH1A1FAAHPRKAA2
SCHEMBL15205904 0.80 GPR119 (0.43) KDM4EALDH1A1HTTHPGDMAPT
SCHEMBL210157 0.80 ALDH1A1 (0.48) KDM4EALDH1A1FAAHLMNAMEN1
SCHEMBL17108787 0.79 SMN1; SMN2 (0.50) KDM4EALDH1A1HTT
SCHEMBL1880665 0.79 SMN1; SMN2 (0.54) KDM4EALDH1A1
SCHEMBL23501608 0.78 ALDH1A1 (0.46) KDM4EALDH1A1HTTMAPTPOLB
SCHEMBL112800 0.78 MC4R (0.47) KDM4EALDH1A1LMNAMAPT
SCHEMBL29934142 0.78 ALDH1A1 (0.46) KDM4EALDH1A1HTTMAPTPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020150545-A1 PYRAZOLE DERIVATIVES AS MODULATORS OF THE WNT/B-CATENIN SIGNALING PATHWAY SAMUMED, LLC (US) 2020-07-23 WO disclosed
EP-2634176-A1 PYRIDINE DERIVATIVE AND MEDICINAL AGENT Nippon Shinyaku Co., Ltd. (JP) 2013-09-04 EP disclosed