SCHEMBL15225276

SCHEMBL15225276

Oc1cc(O)c(-c2n[nH]c3c2CN(Cc2cccc(-n4cccc4)c2)CC3)cc1Cl

nearest known ligand 0.41

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 8/20 0.41
HSP90AB1 P08238 8/20 0.41
MAPK1 P28482 9/20 0.41
MCHR1 Q99705 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15225529 0.92 HSP90AA1 (0.41) HSP90AA1HSP90AB1MAPK1
SCHEMBL2472374 0.91 MAPK1 (0.42) HSP90AA1HSP90AB1MAPK1
SCHEMBL15225020 0.89 HSP90AA1 (0.43) HSP90AA1HSP90AB1MAPK1
SCHEMBL15225169 0.88 HSP90AA1 (0.43) HSP90AA1HSP90AB1MAPK1
SCHEMBL15225644 0.88 LMNA (0.41) HSP90AA1HSP90AB1MAPK1
SCHEMBL15225372 0.88 HSP90AA1 (0.50) HSP90AA1HSP90AB1MAPK1
SCHEMBL15225383 0.87 HSP90AA1 (0.48) HSP90AA1HSP90AB1MAPK1
SCHEMBL2471535 0.85 HSP90AA1 (0.40) HSP90AA1HSP90AB1MAPK1
SCHEMBL15225663 0.83 HSP90AA1 (0.42) HSP90AA1HSP90AB1
SCHEMBL15225304 0.81 DRD2 (0.44) HSP90AA1HSP90AB1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2370437-B1 BICYCLIC PYRAZOLE AND ISOXAZOLE DERIVATIVES AS ANTITUMOR AND ANTINEURODEGENERATIVE AGENTS NERVIANO MEDICAL SCIENCES SRL (IT) 2013-09-04 EP disclosed