SCHEMBL15314734

SCHEMBL15314734

C=C(NNC(=O)OCCc1ccc(N)cc1)OC(C)(C)C

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.42
RAB9A P51151 3/20 0.42
ESRRG P62508 1/20 0.39
MET P08581 2/20 0.38
GAA P10253 1/20 0.36
PPIB P23284 1/20 0.36
PPIA P62937 1/20 0.36
PPID Q08752 1/20 0.36
PPIG Q13427 1/20 0.36
IDO1 P14902 1/20 0.35
EPHX2 P34913 1/20 0.35
CA2 P00918 2/20 0.34
CA1 P00915 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
MAPT P10636 1/20 0.34
GFER P55789 1/20 0.33
ALDH1A1 P00352 1/20 0.33
TP53 P04637 1/20 0.33
GLA P06280 1/20 0.33
CYP3A4 P08684 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL973836 0.89 NPC1 (0.46) NPC1RAB9AESRRGMETGAA
SCHEMBL30479471 0.78 NPC1 (0.46) NPC1RAB9AESRRGMETPPIB
SCHEMBL972841 0.77 NPC1 (0.48) NPC1RAB9AESRRGMETGAA
SCHEMBL27574189 0.77 NPC1 (0.48) NPC1RAB9AESRRGMETPPIB
SCHEMBL15650646 0.75 NPC1 (0.51) NPC1RAB9AESRRGMETPPIB
SCHEMBL30958195 0.74 IDO1 (0.48) ESRRGIDO1CA2CA1SMN1; SMN2
SCHEMBL25266889 0.73 NAAA (0.42) NPC1RAB9ACA2CA1MAPT
SCHEMBL25238911 0.73 NAAA (0.42) NPC1RAB9ACA2CA1MAPT
SCHEMBL448114 0.72 CA2 (0.58) ESRRGIDO1CA2CA1MAPT
SCHEMBL22403769 0.71 GLA (0.51) NPC1RAB9AESRRGMETGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2650287-A1 Thiazole Derivative and use thereof as VAP-1 Inhibitor R-Tech Ueno, Ltd. (JP) 2013-10-16 EP disclosed