SCHEMBL1531740

SCHEMBL1531740

Sc1nnc(-c2cccc3ccccc23)s1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN11 Q06124 1/20 0.47
ALDH1A1 P00352 2/20 0.47
HPGD P15428 2/20 0.47
KDM4E B2RXH2 1/20 0.47
LMNA P02545 1/20 0.47
HSD17B10 Q99714 1/20 0.47
HDAC1 Q13547 1/20 0.45
HDAC2 Q92769 1/20 0.45
ALOX15 P16050 2/20 0.42
DCTPP1 Q9H773 1/20 0.42
HTR2C P28335 5/20 0.41
TGFBR1 P36897 1/20 0.39
MAPT P10636 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
NPC1 O15118 1/20 0.37
CASP3 P42574 1/20 0.37
RAB9A P51151 1/20 0.37
SENP7 Q9BQF6 1/20 0.37
SENP6 Q9GZR1 1/20 0.37
MGAM O43451 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL251035 0.87 KDM4E (0.53) PTPN11ALDH1A1HPGDKDM4ELMNA
SCHEMBL12914313 0.83 PTPN11 (0.50) PTPN11ALDH1A1HPGDKDM4ELMNA
SCHEMBL28827251 0.79 KDM4E (0.61) PTPN11ALDH1A1HPGDKDM4ELMNA
SCHEMBL30987378 0.79 PTPN11 (0.47) PTPN11ALDH1A1HPGDKDM4ELMNA
SCHEMBL27646939 0.77 GUSB (0.49) PTPN11ALDH1A1HPGDKDM4ELMNA
SCHEMBL27639574 0.76 GUSB (0.48) PTPN11ALDH1A1HPGDKDM4ELMNA
SCHEMBL17819129 0.76 ALOX15 (0.54) PTPN11ALDH1A1HPGDKDM4ELMNA
SCHEMBL27620753 0.76 GUSB (0.51) PTPN11ALDH1A1HPGDKDM4ELMNA
SCHEMBL968101 0.76 KDM4E (0.61) ALDH1A1HPGDKDM4EHSD17B10DCTPP1
SCHEMBL1107963 0.75 KDM4E (0.47) PTPN11ALDH1A1HPGDKDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011028651-A1 INHIBITORS OF HUMAN 15-LIPOXYGENASE-1 THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2011-03-10 WO disclosed
US-6080772-A 2-AMINOTHIAZOLE TRIAZOLE OR TETRAZOLE COMPOUND FOR REGULATING PROTEIN TYROSINE PHOSPHATASE ACTIVITY SUGEN, INC. (US) 2000-06-27 US disclosed