SCHEMBL15319487

SCHEMBL15319487

O=Cc1cccc(-c2ccc[nH]2)c1Cl

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKA O14965 1/20 0.41
KDR P35968 1/20 0.41
MEN1 O00255 3/20 0.35
KMT2A Q03164 3/20 0.35
LMNA P02545 2/20 0.35
TDP1 Q9NUW8 2/20 0.35
THRB P10828 1/20 0.35
BLM P54132 1/20 0.35
CYP1A1 P04798 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2D6 P10635 1/20 0.33
MAPT P10636 1/20 0.33
AHR P35869 1/20 0.33
CYP1B1 Q16678 1/20 0.33
ERN1 O75460 2/20 0.32
CNR1 P21554 1/20 0.32
ALDH1A1 P00352 2/20 0.31
CHRNB4 P30926 1/20 0.31
CHRNA3 P32297 1/20 0.31
PARP1 P09874 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30239797 0.82 MEN1 (0.46) AURKAKDRMEN1KMT2ALMNA
SCHEMBL5961899 0.82 MEN1 (0.46) AURKAKDRMEN1KMT2ALMNA
SCHEMBL10702785 0.76 AURKA (0.42) AURKAKDRMEN1KMT2ABLM
SCHEMBL31190899 0.76 IDO1 (0.54)
SCHEMBL3794351 0.72 TDP1 (0.58) MEN1KMT2ALMNATDP1THRB
SCHEMBL4033813 0.71 KMT2A (0.46) MEN1KMT2ALMNATDP1THRB
SCHEMBL10533687 0.71 TDP1 (0.46) MEN1KMT2ALMNATDP1THRB
SCHEMBL3936518 0.68 ALDH1A1 (0.50) MEN1KMT2ALMNATDP1THRB
SCHEMBL18519466 0.68 ALDH1A1 (0.48) AURKAKDRMEN1KMT2AMAPT
SCHEMBL15416821 0.68 KDR (0.47) AURKAKDRPARP1CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2833879-A1 KYNURENINE-3-MONOOXYGENASE INHIBITORS, PHARMACEUTICAL COMPOSITIONS, AND METHODS OF USE THEREOF CHDI Foundation, Inc. (US) 2015-02-11 EP disclosed
WO-2013151707-A1 KYNURENINE-3-MONOOXYGENASE INHIBITORS, PHARMACEUTICAL COMPOSITIONS, AND METHODS OF USE THEREOF CHDI FOUNDATION, INC. (US) 2013-10-10 WO disclosed