SCHEMBL15327461

SCHEMBL15327461

N#CC1(NC(=O)O[C@H]2C[C@@H](S(=O)(=O)c3ccc(-n4cccn4)cc3Cl)CN2C(=O)C2(c3ccc(Cl)cc3)CC2)CC1

nearest known ligand 0.58

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CTSL P07711 14/20 0.58
CTSS P25774 16/20 0.51
CTSK P43235 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15327336 0.93 CTSS (0.50) CTSLCTSSCTSK
SCHEMBL696735 0.90 CTSL (0.73) CTSLCTSSCTSK
SCHEMBL15327642 0.88 CTSS (0.54) CTSLCTSSCTSK
SCHEMBL15327317 0.88 CTSL (0.56) CTSLCTSSCTSK
SCHEMBL15327591 0.88 CTSL (0.66) CTSLCTSSCTSK
SCHEMBL15327480 0.87 CTSL (0.57) CTSLCTSSCTSK
SCHEMBL15327152 0.87 CTSS (0.66) CTSS
SCHEMBL15327265 0.87 CTSS (0.66) CTSS
SCHEMBL15327468 0.87 CTSL (0.59) CTSLCTSSCTSK
SCHEMBL15327466 0.86 CTSL (0.53) CTSLCTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2421826-B1 PROLINE DERIVATIVES AS CATHEPSIN INHIBITORS HOFFMANN LA ROCHE (CH) 2013-10-23 EP claimed