Mexenone

Mexenone

SCHEMBL15327784

COc1ccc(C(=O)c2ccc(C)cc2)c(O)c1.COc1ccc(C(=O)c2ccccc2O)c(O)c1

nearest known ligand 0.78

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 4/20 0.78
LMNA P02545 3/20 0.78
CYP1A2 P05177 2/20 0.78
PGR P06401 2/20 0.78
SLC6A2 P23975 2/20 0.78
CYP2C19 P33261 2/20 0.78
CYP3A4 P08684 2/20 0.78
ADORA3 P0DMS8 1/20 0.78
AR P10275 1/20 0.78
CHRM1 P11229 1/20 0.78
ALOX15 P16050 1/20 0.78
TBXA2R P21731 1/20 0.78
ADRA1A P35348 1/20 0.78
HIF1A Q16665 1/20 0.78
ALDH1A1 P00352 4/20 0.72
HTT P42858 3/20 0.72
MAPK1 P28482 2/20 0.72
CYP2D6 P10635 1/20 0.72
PDE4A P27815 1/20 0.72
HRH1 P35367 1/20 0.72

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Mexenone SCHEMBL4595243 0.92 HPGD (0.66) HPGDLMNACYP1A2PGRSLC6A2
Mexenone SCHEMBL6847100 0.92 LMNA (0.86) HPGDLMNACYP1A2PGRSLC6A2
Mexenone SCHEMBL8017506 0.92 LMNA (0.74) HPGDLMNACYP1A2PGRSLC6A2
Mexenone SCHEMBL29365598 0.92 LMNA (0.74) HPGDLMNACYP1A2PGRSLC6A2
Mexenone SCHEMBL39448 0.92 LMNA (0.74) HPGDLMNACYP1A2PGRSLC6A2
Dioxybenzone SCHEMBL5161579 0.90 HPGD (0.88) HPGDLMNACYP1A2PGRSLC6A2
Dioxybenzone SCHEMBL28167789 0.90 HPGD (0.85) HPGDLMNACYP1A2PGRSLC6A2
Dioxybenzone SCHEMBL4923214 0.90 HPGD (0.88) HPGDLMNACYP1A2PGRSLC6A2
Mexenone SCHEMBL29612353 0.90 LMNA (0.72) HPGDLMNACYP1A2PGRSLC6A2
Oxybenzone SCHEMBL28230340 0.89 HPGD (0.91) HPGDLMNACYP1A2PGRSLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 26 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4157213-A1 SUNSCREEN WITH A COMBINATION OF CARNAUBA WAX AND HYDROGENATED RAPESEED OIL Beiersdorf AG (DE) 2023-04-05 EP claimed
EP-4037642-A1 NOVEL SUN PROTECTIVE AGENT CONTAINING BISMUTH OXYCHLORIDE FOR PROTECTION AGAINST BLUE LIGHT Beiersdorf AG (DE) 2022-08-10 EP claimed
EP-3923900-A1 ODOR-STABLE ETHANOLIC PREPARATION CONTAINING OCTOCRYLENE Beiersdorf AG (DE) 2021-12-22 EP claimed
WO-2021239385-A1 SUNSCREEN WITH A COMBINATION OF CARNAUBA WAX AND HYDROGENATED RAPESEED OIL BEIERSDORF AG (DE) 2021-12-02 WO claimed
WO-2021063609-A1 BISMUTH OXYCHLORIDE-CONTAINING SUNSCREEN FOR PROTECTION FROM BLUE LIGHT BEIERSDORF AG (DE) 2021-04-08 WO claimed
WO-2021063610-A1 NOVEL SUN PROTECTIVE AGENT CONTAINING BISMUTH OXYCHLORIDE FOR PROTECTION AGAINST BLUE LIGHT BEIERSDORF AG (DE) 2021-04-08 WO claimed
WO-2020164905-A1 ODOR-STABLE ETHANOLIC PREPARATION CONTAINING OCTOCRYLENE BEIERSDORF AG (DE) 2020-08-20 WO claimed
EP-3137042-B2 SUNSCREEN HAVING REDUCED TENDENCY TO STAIN TEXTILES II BEIERSDORF AG (DE) 2024-06-26 EP disclosed
EP-4157213-A1 SUNSCREEN WITH A COMBINATION OF CARNAUBA WAX AND HYDROGENATED RAPESEED OIL Beiersdorf AG (DE) 2023-04-05 EP disclosed
WO-2023046568-A1 COSMETIC PREPARATION CONTAINING LIME GLASS BEADS WITH HIGH SPECIFIC WEIGHT BEIERSDORF AG (DE) 2023-03-30 WO disclosed
EP-3137041-B2 SUNSCREEN HAVING REDUCED TENDENCY TO STAIN TEXTILES BEIERSDORF AG (DE) 2023-01-18 EP disclosed
EP-4103148-A1 POLYACRYLATE-FREE COSMETIC PREPARATION Beiersdorf AG (DE) 2022-12-21 EP disclosed
EP-4096794-A1 SUNSCREEN WITH PIGMENT FILTER SEPARATION Beiersdorf AG (DE) 2022-12-07 EP disclosed
WO-2021151694-A1 SUNSCREEN WITH PIGMENT FILTER SEPARATION BEIERSDORF AG (DE) 2021-08-05 WO disclosed
WO-2021063609-A1 BISMUTH OXYCHLORIDE-CONTAINING SUNSCREEN FOR PROTECTION FROM BLUE LIGHT BEIERSDORF AG (DE) 2021-04-08 WO disclosed
WO-2021063610-A1 NOVEL SUN PROTECTIVE AGENT CONTAINING BISMUTH OXYCHLORIDE FOR PROTECTION AGAINST BLUE LIGHT BEIERSDORF AG (DE) 2021-04-08 WO disclosed
WO-2021043721-A1 USE OF COSMETIC PREPARATIONS FOR IMPROVING THE VISIBILITY OF SUBEPIDERMAL PIGMENTS BEIERSDORF AG (DE) 2021-03-11 WO disclosed
EP-3687630-A1 COSMETIC PREPARATION CONTAINING CETYL-DIGLYCERYL TRIS(TRIMETHYLSILOXY)SILYLETHYL DIMETHICONE Beiersdorf AG (DE) 2020-08-05 EP disclosed
EP-3173129-B1 SUNSCREEN COMPRISING TITANIUM DIOXIDE AND ETHYLHEXYL SALICYLATE BEIERSDORF AG (DE) 2020-01-29 EP disclosed
EP-2099424-B1 COSMETIC FORMULATION CONTAINING GLUCOSYL GLYCERIDES AND SKIN LIGHTENING AGENTS BEIERSDORF AG (DE) 2013-10-23 EP disclosed