SCHEMBL15329664

SCHEMBL15329664

COCCC(C)(Oc1cccc(C=O)c1)C(=O)O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SRC P12931 1/20 0.43
MAOB P27338 6/20 0.42
MAOA P21397 5/20 0.42
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
TDP1 Q9NUW8 1/20 0.41
UNG P13051 1/20 0.41
ALDH1A1 P00352 2/20 0.41
POLB P06746 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.39
KDM4E B2RXH2 2/20 0.39
GAA P10253 1/20 0.39
MAPT P10636 1/20 0.39
HPGD P15428 1/20 0.39
KMT2A Q03164 1/20 0.39
FOS P01100 1/20 0.39
JUN P05412 1/20 0.39
BCHE P06276 1/20 0.39
PPARA Q07869 2/20 0.37
TRIM24 O15164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2556213 0.87 MAOA (0.43) SRCMAOBMAOANPC1RAB9A
SCHEMBL15329910 0.87 SMN1; SMN2 (0.44) SRCMAOBMAOANPC1RAB9A
SCHEMBL2562722 0.84 ALDH1A1 (0.42) ALDH1A1KMT2APPARA
SCHEMBL2554985 0.84 PPARG (0.48) SRCMAOBMAOANPC1RAB9A
SCHEMBL2553855 0.84 MAOA (0.41) SRCMAOBMAOANPC1RAB9A
SCHEMBL2559935 0.81 MAOA (0.43) SRCMAOBMAOANPC1RAB9A
SCHEMBL2559049 0.81 MAOB (0.47) MAOBMAOANPC1RAB9AALDH1A1
SCHEMBL2174559 0.78 PPARA (0.51) SRCMAOBMAOAUNGALDH1A1
SCHEMBL2557997 0.78 LMNA (0.39) NPC1RAB9AALDH1A1POLBSMN1; SMN2
SCHEMBL3066417 0.75 SRC (0.46) SRCMAOBMAOANPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220340893-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2022-10-27 US disclosed
US-11225655-B2 Bi-functional complexes and methods for making and using such complexes NUEVOLUTION A/S (DK) 2022-01-18 US disclosed
EP-3540059-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES Nuevolution A/S (DK) 2019-09-18 EP disclosed
EP-2558577-B1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION AS (DK) 2018-12-12 EP disclosed
US-20130281324-A1 BI-FUNCTINAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2013-10-24 US disclosed