SCHEMBL15330774

SCHEMBL15330774

NC(=O)CC1CCN(CCC=O)CC1

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.35
POLB P06746 1/20 0.33
HTT P42858 1/20 0.33
GNAI3 P08754 2/20 0.32
GNAO1 P09471 2/20 0.32
GNAI1 P63096 2/20 0.32
DRD2 P14416 2/20 0.32
HTR2A P28223 2/20 0.32
HTR2C P28335 2/20 0.32
HTR2B P41595 2/20 0.32
SIGMAR1 Q99720 2/20 0.32
EPHX1 P07099 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26049827 0.82 CHRM1 (0.39) L3MBTL1SMN1; SMN2POLBHTTGNAI3
SCHEMBL22266364 0.81 SLC18A3 (0.40) LTA4HL3MBTL1SMN1; SMN2POLBHTT
SCHEMBL2556227 0.81 LTA4H (0.39) LTA4HSMN1; SMN2DRD2HTR2AHTR2C
SCHEMBL27897215 0.80 SIGMAR1 (0.33) POLBHTTGNAI3GNAO1GNAI1
SCHEMBL22266187 0.80 L3MBTL1 (0.55) LTA4HL3MBTL1SMN1; SMN2POLBSIGMAR1
SCHEMBL2563207 0.80 SMN1; SMN2 (0.56) LTA4HL3MBTL1SMN1; SMN2POLB
SCHEMBL18666615 0.79 LTA4H (0.37) LTA4HGNAI3GNAO1GNAI1SIGMAR1
SCHEMBL23349993 0.79 HTT (0.51) LTA4HL3MBTL1SMN1; SMN2POLBHTT
SCHEMBL22266266 0.77 ANPEP (0.38) LTA4HL3MBTL1SMN1; SMN2POLBGNAO1
SCHEMBL8186300 0.77 SMN1; SMN2 (0.39) SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220340893-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2022-10-27 US disclosed
US-11225655-B2 Bi-functional complexes and methods for making and using such complexes NUEVOLUTION A/S (DK) 2022-01-18 US disclosed
EP-3540059-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES Nuevolution A/S (DK) 2019-09-18 EP disclosed
EP-2558577-B1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION AS (DK) 2018-12-12 EP disclosed
US-20130281324-A1 BI-FUNCTINAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2013-10-24 US disclosed