SCHEMBL15415976

SCHEMBL15415976

COc1cc(N2CCOC2)ccc1Br

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 6/20 0.46
MEN1 O00255 5/20 0.46
THRB P10828 2/20 0.46
MAPT P10636 8/20 0.45
ALDH1A1 P00352 7/20 0.45
GAA P10253 3/20 0.45
MAPK1 P28482 2/20 0.45
HPGD P15428 3/20 0.43
POLB P06746 1/20 0.43
HTT P42858 2/20 0.43
GRM2 Q14416 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
PTPN1 P18031 1/20 0.42
HIF1A Q16665 1/20 0.42
TGFBR1 P36897 1/20 0.41
ACVR1 Q04771 1/20 0.41
KDM4E B2RXH2 4/20 0.41
CYP3A4 P08684 1/20 0.41
TSHR P16473 1/20 0.41
CYP2C19 P33261 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30602381 0.91 MEN1 (0.54) KMT2AMEN1THRBMAPTALDH1A1
SCHEMBL807233 0.91 MEN1 (0.54) KMT2AMEN1THRBMAPTALDH1A1
SCHEMBL23705839 0.79 ALDH1A1 (0.55) KMT2AMEN1MAPTALDH1A1MAPK1
SCHEMBL31091978 0.79 ALDH1A1 (0.55) KMT2AMEN1MAPTALDH1A1MAPK1
SCHEMBL2498472 0.78 MAPT (0.63) KMT2AMEN1THRBMAPTALDH1A1
SCHEMBL807418 0.78 ALDH1A1 (0.58) KMT2AMEN1MAPTALDH1A1PTPN1
SCHEMBL5528296 0.76 MAPK1 (0.49) KMT2AMEN1MAPTALDH1A1MAPK1
SCHEMBL2384047 0.76 SIRT6 (0.58) KMT2AMEN1MAPTALDH1A1GAA
SCHEMBL19500869 0.76 HIF1A (0.62) KMT2AMEN1THRBMAPTALDH1A1
SCHEMBL255446 0.75 CHRNB2 (0.60) MAPTTGFBR1ACVR1CYP2C19LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2872506-A1 METHOD FOR PREPARING SUBSTITUTED TRIAZOLOPYRIDINES Bayer Pharma Aktiengesellschaft (DE) 2015-05-20 EP disclosed
WO-2014009219-A1 METHOD FOR PREPARING SUBSTITUTED TRIAZOLOPYRIDINES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2014-01-16 WO disclosed