SCHEMBL15417779

SCHEMBL15417779

CNC(=O)c1cc(C)c(C)cn1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.47
RAB9A P51151 3/20 0.47
MAPT P10636 3/20 0.47
KDM4E B2RXH2 1/20 0.47
ALDH1A1 P00352 1/20 0.47
LMNA P02545 1/20 0.47
TP53 P04637 1/20 0.47
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2C9 P11712 1/20 0.47
PKM P14618 1/20 0.47
HPGD P15428 1/20 0.47
TSHR P16473 1/20 0.47
APEX1 P27695 1/20 0.47
CYP2C19 P33261 1/20 0.47
THPO P40225 1/20 0.47
PMP22 Q01453 1/20 0.47
HSD17B10 Q99714 1/20 0.47
BAZ2B Q9UIF8 1/20 0.47
CNR1 P21554 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1459777 0.85 NPC1 (0.43) NPC1RAB9AMAPTKDM4EALDH1A1
SCHEMBL23618778 0.85 UHRF1 (0.47) NPC1RAB9AMAPTKDM4EALDH1A1
SCHEMBL30992044 0.85 UHRF1 (0.47) NPC1RAB9AMAPTKDM4EALDH1A1
SCHEMBL23343417 0.85 MAPT (0.43) NPC1RAB9AMAPTKDM4EALDH1A1
SCHEMBL30108322 0.83 MAPT (0.42) NPC1RAB9AMAPTKDM4EALDH1A1
SCHEMBL15417325 0.83 RAB9A (0.42) NPC1RAB9AMAPTKDM4EALDH1A1
SCHEMBL17553883 0.83 NOS3 (0.49) NPC1RAB9AMAPTKDM4EALDH1A1
SCHEMBL24956360 0.82 HPGDS (0.43) NPC1RAB9AMAPTKDM4EALDH1A1
SCHEMBL30108286 0.82 MAPT (0.41) NPC1RAB9AMAPTKDM4EALDH1A1
SCHEMBL19249055 0.81 BAZ2B (0.42) NPC1RAB9AMAPTKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2651899-B1 SUBSTITUTED 6,6-FUSED NITROGENOUS HETEROCYCLIC COMPOUNDS AND USES THEREOF HOFFMANN LA ROCHE (CH) 2017-05-31 EP disclosed
US-8623889-B2 Substituted 6,6-fused nitrogenous heterocyclic compounds and uses thereof GENENTECH, INC. (US) 2014-01-07 US disclosed