SCHEMBL15427263

SCHEMBL15427263

O=C(CI)NCC1(O)CCC1

nearest known ligand 0.33

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.33
P2RX7 Q99572 18/20 0.33
LMNA P02545 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22259417 0.79 ALDH1A1 (0.41) BRD4P2RX7
SCHEMBL15427281 0.79 MEN1 (0.41) BRD4P2RX7LMNA
SCHEMBL15621584 0.76 LMNA (0.56) BRD4P2RX7LMNA
SCHEMBL19116500 0.76 SMN1; SMN2 (0.42) BRD4P2RX7LMNA
SCHEMBL28521208 0.76 P2RX7 (0.39) BRD4P2RX7
SCHEMBL19151155 0.75 LMNA (0.42) BRD4P2RX7LMNA
SCHEMBL22449838 0.75 ALDH1A1 (0.41) BRD4P2RX7LMNA
SCHEMBL15617686 0.75 HPGD (0.37) BRD4P2RX7LMNA
SCHEMBL15932513 0.74 ALDH1A1 (0.39) BRD4P2RX7
SCHEMBL20888086 0.74 TSHR (0.45) BRD4P2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2870153-B1 SULFONYL CONTAINING BENZOTHIAZOLE INHIBITORS OF ENDOTHELIAL LIPASE BRISTOL MYERS SQUIBB CO (US) 2016-11-02 EP disclosed
WO-2014011513-A1 SULFONYL CONTAINING BENZOTHIAZOLE INHIBITORS OF ENDOTHELIAL LIPASE BRISTOL-MYERS SQUIBB COMPANY (US) 2014-01-16 WO disclosed