SCHEMBL15428705

SCHEMBL15428705

Cc1ccc(Nc2ncc3cnn([C@H]4CC[C@H](NC(=O)O)CC4)c3n2)cc1S(N)(=O)=O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 19/20 0.48
AURKA O14965 18/20 0.48
CCNB1 P14635 12/20 0.48
AURKB Q96GD4 6/20 0.47
CDK2 P24941 2/20 0.42
CDK9 P50750 1/20 0.42
TTK P33981 1/20 0.42
PLK4 O00444 1/20 0.42
PDPK1 O15530 1/20 0.42
DAPK3 O43293 1/20 0.42
JAK2 O60674 1/20 0.42
MAP4K4 O95819 1/20 0.42
PAK4 O96013 1/20 0.42
CHEK2 O96017 1/20 0.42
EGFR P00533 1/20 0.42
ERBB2 P04626 1/20 0.42
NTRK1 P04629 1/20 0.42
PRKCG P05129 1/20 0.42
INSR P06213 1/20 0.42
LCK P06239 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15428704 1.00 CDK1 (0.48) CDK1AURKACCNB1AURKBCDK2
SCHEMBL10167379 0.90 CDK1 (0.44) CDK1AURKACCNB1AURKBCDK2
SCHEMBL343351 0.90 CDK1 (0.44) CDK1AURKACCNB1AURKBCDK2
SCHEMBL342357 0.88 AURKA (0.52) CDK1AURKACCNB1AURKB
SCHEMBL10167410 0.88 AURKA (0.52) CDK1AURKACCNB1AURKB
SCHEMBL342650 0.85 CDK1 (0.46) CDK1AURKACCNB1AURKBCDK2
SCHEMBL342651 0.85 CDK1 (0.46) CDK1AURKACCNB1AURKBCDK2
SCHEMBL343811 0.85 AURKA (0.51) CDK1AURKACCNB1AURKBCDK2
SCHEMBL342652 0.84 CDK1 (0.48) CDK1AURKACCNB1AURKBCDK2
SCHEMBL343675 0.82 CCND3 (0.51) CDK1AURKACCNB1AURKBCDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8637529-B2 Pyrazolo[3,4-d]pyrimidine compounds AbbYie Inc. (US) 2014-01-28 US disclosed