SCHEMBL343351

SCHEMBL343351

Cc1ccc(Nc2ncc3cnn(C4CCC(NC(=O)OC(C)(C)C)CC4)c3n2)cc1S(N)(=O)=O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 16/20 0.44
AURKA O14965 15/20 0.44
CCNB1 P14635 9/20 0.44
AURKB Q96GD4 6/20 0.44
TTK P33981 2/20 0.42
CDK4 P11802 1/20 0.42
CCND1 P24385 1/20 0.42
CCND2 P30279 1/20 0.42
CCND3 P30281 1/20 0.42
RET P07949 2/20 0.41
CDK2 P24941 2/20 0.41
PLK4 O00444 1/20 0.41
PDPK1 O15530 1/20 0.41
DAPK3 O43293 1/20 0.41
JAK2 O60674 1/20 0.41
MAP4K4 O95819 1/20 0.41
PAK4 O96013 1/20 0.41
CHEK2 O96017 1/20 0.41
EGFR P00533 1/20 0.41
ERBB2 P04626 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10167379 1.00 CDK1 (0.44) CDK1AURKACCNB1AURKBTTK
SCHEMBL15428704 0.90 CDK1 (0.48) CDK1AURKACCNB1AURKBTTK
SCHEMBL15428705 0.90 CDK1 (0.48) CDK1AURKACCNB1AURKBTTK
SCHEMBL10167369 0.88 SYK (0.40) CDK1AURKAAURKBTTKCDK4
SCHEMBL343675 0.86 CCND3 (0.51) CDK1AURKACCNB1AURKBCDK4
SCHEMBL342357 0.84 AURKA (0.52) CDK1AURKACCNB1AURKB
SCHEMBL10167410 0.84 AURKA (0.52) CDK1AURKACCNB1AURKB
SCHEMBL343811 0.83 AURKA (0.51) CDK1AURKACCNB1AURKBCDK4
SCHEMBL342650 0.81 CDK1 (0.46) CDK1AURKACCNB1AURKBRET
SCHEMBL342651 0.81 CDK1 (0.46) CDK1AURKACCNB1AURKBRET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8637529-B2 Pyrazolo[3,4-d]pyrimidine compounds AbbYie Inc. (US) 2014-01-28 US claimed
US-20120015963-A1 NOVEL PYRAZOLO[3,4-d]PYRIMIDINE COMPOUNDS ABBOTT LABORATORIES (US) 2012-01-19 US claimed
US-8637529-B2 Pyrazolo[3,4-d]pyrimidine compounds AbbYie Inc. (US) 2014-01-28 US disclosed
US-20120015963-A1 NOVEL PYRAZOLO[3,4-d]PYRIMIDINE COMPOUNDS ABBOTT LABORATORIES (US) 2012-01-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120015963-A1 NOVEL PYRAZOLO[3,4-d]PYRIMIDINE COMPOUNDS CHUK, MAP2K2, CDK3 CDK1 10/4885AURKA 784/4885CCNB1 388/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.